Compile Data Set for Download or QSAR
maximum 50k data
Found 50 with Last Name = 'matsuda' and Initial = 'f'
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180193(AZD-2624 | AZD2624)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180171(CHEMBL3813763)
Affinity DataIC50:  3.90nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180169(CHEMBL3814787)
Affinity DataIC50:  5.60nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180174(CHEMBL3813719)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)
Affinity DataIC50:  8.40nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50299467((5S,8S,14S,17S,20S,23S,26S,29S,32S)-26-((1H-imidaz...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028014(CHEMBL3361397)
Affinity DataIC50:  22nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180170(CHEMBL3815065)
Affinity DataIC50:  24nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028015(CHEMBL3361398)
Affinity DataIC50:  43nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180175(CHEMBL3813835)
Affinity DataIC50:  44nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028021(CHEMBL3361404)
Affinity DataIC50:  56nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataIC50:  56nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028016(CHEMBL3361399)
Affinity DataIC50:  59nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180168(CHEMBL3814967)
Affinity DataIC50:  154nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180172(CHEMBL3813735)
Affinity DataIC50:  245nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028025(CHEMBL3361408)
Affinity DataIC50:  360nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180173(CHEMBL3815072)
Affinity DataIC50:  390nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180176(CHEMBL3814793)
Affinity DataIC50:  965nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028024(CHEMBL3361407)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180184(CHEMBL3813742)
Affinity DataIC50:  1.53E+3nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028018(CHEMBL3361401)
Affinity DataIC50:  2.30E+3nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028017(CHEMBL3361400)
Affinity DataIC50:  2.90E+3nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180166(CHEMBL3814985)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180167(CHEMBL3815160)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028023(CHEMBL3361406)
Affinity DataIC50:  1.30E+4nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028022(CHEMBL3361405)
Affinity DataIC50:  1.90E+4nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028020(CHEMBL3361403)
Affinity DataIC50: >1.00E+7nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028019(CHEMBL3361402)
Affinity DataIC50: >1.00E+7nMAssay Description:Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391540(CHEMBL2147469)
Affinity DataEC50:  200nMAssay Description:Inhibition of cathepsin B using Z-Phe-Arg-MCA as substrate incubated for 10 mins prior to substrate addition measured after 30 mins by fluorimetric a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391540(CHEMBL2147469)
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391541(CHEMBL2147467)
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of bovine thrombin using Bz-Phe-Val-Arg-pNA as substrate incubated for 5 mins prior to substrate addition measured after 30 mins by fluori...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391540(CHEMBL2147469)
Affinity DataEC50:  7.50E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391540(CHEMBL2147469)
Affinity DataEC50:  2.10E+3nMAssay Description:Inhibition of bovine thrombin using Bz-Phe-Val-Arg-pNA as substrate incubated for 5 mins prior to substrate addition measured after 30 mins by fluori...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028021(CHEMBL3361404)
Affinity DataEC50:  19nMAssay Description:Agonist activity at rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028025(CHEMBL3361408)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028024(CHEMBL3361407)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028023(CHEMBL3361406)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391541(CHEMBL2147467)
Affinity DataEC50:  700nMAssay Description:Inhibition of cathepsin B using Z-Phe-Arg-MCA as substrate incubated for 10 mins prior to substrate addition measured after 30 mins by fluorimetric a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028021(CHEMBL3361404)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028020(CHEMBL3361403)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028019(CHEMBL3361402)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028018(CHEMBL3361401)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028017(CHEMBL3361400)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028016(CHEMBL3361399)
Affinity DataEC50:  91nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028015(CHEMBL3361398)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028014(CHEMBL3361397)
Affinity DataEC50:  330nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50299467((5S,8S,14S,17S,20S,23S,26S,29S,32S)-26-((1H-imidaz...)
Affinity DataEC50:  64nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50028022(CHEMBL3361405)
Affinity DataEC50:  920nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed