Affinity DataKi: <1nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to Cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to reninMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to reninMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to Cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Tested for the inhibition of HIV-2 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 33nM ΔG°: -44.4kJ/mole IC50: 58nMpH: 4.7 T: 2°CAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of HIV-1 protease in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to Cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Compound was evaluated for the inhibition of HIV-2 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Evaluated for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair