TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.240nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.530nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.550nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.580nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.580nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.580nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.580nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.610nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
Affinity DataIC50: 0.640nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.710nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.760nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.760nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.890nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Agonistic activity towards Opioid receptor delta 1 was determined by evaluating the inhibitory activity towards electrically stimulated mouse vas def...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 8.90nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Inhibition of binding [3H]-DAMGO at Opioid receptor mu 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 in guinea pig brain using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair