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Found 176 with Last Name = 'meyer' and Initial = 'jp'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033139(CHEMBL2370495 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*...)
Affinity DataIC50:  0.240nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038019(CHEMBL411338 | Tyr-Gly-Gly-Phe-D-Leu-Arg-Arg-Ile-A...)
Affinity DataIC50:  0.530nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453783(CHEMBL2311023)
Affinity DataIC50:  0.550nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataIC50:  0.580nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033143(CHEMBL216640 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...)
Affinity DataIC50:  0.580nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataIC50:  0.580nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036267(CHEMBL268874 | Dyn A(H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  0.580nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453785(CHEMBL2311025)
Affinity DataIC50:  0.610nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453785(CHEMBL2311025)
Affinity DataIC50:  0.640nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038020(CHEMBL2370618 | Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-...)
Affinity DataIC50:  0.710nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50138774(CHEMBL415795 | Linear [D-Ala3]Dyn A-(1-11)NH2)
Affinity DataIC50:  0.760nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051599(CHEMBL415224 | Dynorphin A analogues)
Affinity DataIC50:  0.760nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051595(CHEMBL413228 | Dynorphin A analogues)
Affinity DataIC50:  0.890nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453782(CHEMBL2370497)
Affinity DataIC50:  0.900nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038016(CHEMBL2370611 | Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-...)
Affinity DataIC50:  1nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453445(CHEMBL2112652)
Affinity DataIC50:  1nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036266(CHEMBL262963 | Dyn A(H-Tyr-Gly-Ala-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  1.10nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038012(CHEMBL2370629 | Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-...)
Affinity DataIC50:  1.10nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051594(CHEMBL407303 | Dynorphin A analogues)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038014(CHEMBL2370622 | Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Ar...)
Affinity DataIC50:  2nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038010(CHEMBL2370627 | Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Ar...)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038011(CHEMBL2370612 | Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Ar...)
Affinity DataIC50:  3.10nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033142(CHEMBL2370496 | H-Tyr-Gly-Gly-Phe-Leu-Lys*-Arg*-Il...)
Affinity DataIC50:  4nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033142(CHEMBL2370496 | H-Tyr-Gly-Gly-Phe-Leu-Lys*-Arg*-Il...)
Affinity DataIC50:  4nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038014(CHEMBL2370622 | Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Ar...)
Affinity DataIC50:  5nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038019(CHEMBL411338 | Tyr-Gly-Gly-Phe-D-Leu-Arg-Arg-Ile-A...)
Affinity DataIC50:  5.20nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038020(CHEMBL2370618 | Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-...)
Affinity DataIC50:  5.20nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033139(CHEMBL2370495 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*...)
Affinity DataIC50:  5.20nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051603(CHEMBL412792 | Dynorphin A analogues)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051592(CHEMBL2369902 | [(2S,3R)-beta-MePhe3] Dynorphin A ...)
Affinity DataIC50:  6nMAssay Description:Agonistic activity towards Opioid receptor delta 1 was determined by evaluating the inhibitory activity towards electrically stimulated mouse vas def...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051592(CHEMBL2369902 | [(2S,3R)-beta-MePhe3] Dynorphin A ...)
Affinity DataIC50:  6nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038010(CHEMBL2370627 | Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Ar...)
Affinity DataIC50:  7.10nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453784(CHEMBL2311024)
Affinity DataIC50:  8nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50454203(CHEMBL2369896)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453782(CHEMBL2370497)
Affinity DataIC50:  9nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033141(CHEMBL2370494 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...)
Affinity DataIC50:  9.20nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of binding [3H]-DAMGO at Opioid receptor mu 1 of guinea pig brain membrane (GPB) homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036267(CHEMBL268874 | Dyn A(H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  9.90nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 in guinea pig brain using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033143(CHEMBL216640 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...)
Affinity DataIC50:  9.90nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataIC50:  9.90nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453783(CHEMBL2311023)
Affinity DataIC50:  12nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453445(CHEMBL2112652)
Affinity DataIC50:  12nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033142(CHEMBL2370496 | H-Tyr-Gly-Gly-Phe-Leu-Lys*-Arg*-Il...)
Affinity DataIC50:  13nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453445(CHEMBL2112652)
Affinity DataIC50:  14nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038007(CHEMBL2370626 | Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Ar...)
Affinity DataIC50:  15nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038013(CHEMBL374268 | Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg...)
Affinity DataIC50:  15nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038020(CHEMBL2370618 | Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-...)
Affinity DataIC50:  16nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033141(CHEMBL2370494 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...)
Affinity DataIC50:  17nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50038016(CHEMBL2370611 | Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-...)
Affinity DataIC50:  17nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033141(CHEMBL2370494 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...)
Affinity DataIC50:  17nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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