Affinity DataKi: 0.110nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonistic activity against orphan FQ receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonistic activity against orphan FQ receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Antagonistic activity against orphan FQ receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Agonist activity as stimulation of [35S]-GTP-gamma binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Agonist activity as stimulation of [35S]-GTP-gamma binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Antagonistic activity against orphan FQ receptorMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity for opioid receptor like 1 expressed in HEK-293 cells More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Antagonistic activity against orphan FQ receptorMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Antagonistic activity against orphan FQ receptorMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Binding affinity for recombinant human mu-opioid receptor was determined by using [3H]- diprenophine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Antagonistic activity against orphan FQ receptorMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Binding affinity for opioid receptor like 1 expressed in HEK-293 cells More data for this Ligand-Target Pair