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Found 23 with Last Name = 'moore' and Initial = 'ja'
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50:  0.0440nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248496(2-(4-(2-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-indol...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248450(2-(4-fluorophenyl)-6-(piperidin-4-yl)-3-(pyridin-4...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248451(2-(4-fluorophenyl)-6-(1-methylpiperidin-4-yl)-3-(p...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248452(6-(1-ethylpiperidin-4-yl)-2-(4-fluorophenyl)-3-(py...)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248396(4-(2-(4-fluorophenyl)-6-(piperidin-4-yl)-1H-indol-...)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248543(4-(2-(4-fluorophenyl)-6-(1-methylpiperidin-4-yl)-1...)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248397(2-(4-(3-(2-aminopyrimidin-4-yl)-2-(4-fluorophenyl)...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248399(2-(4-fluorophenyl)-6-(1-methylpiperidin-4-yl)-3-(p...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248498(2-(4-fluorophenyl)-6-(1-methylazetidin-3-yl)-3-(py...)
Affinity DataIC50:  0.620nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248398(2-(4-fluorophenyl)-6-(piperidin-4-yl)-3-(pyrimidin...)
Affinity DataIC50:  0.650nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248449(2-(4-(2-(4-fluorophenyl)-3-(pyrimidin-4-yl)-1H-ind...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248499(2-(4-fluorophenyl)-6-((1-methylpiperidin-4-yl)meth...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248542(2-(4-fluorophenyl)-6-((4-methylpiperazin-1-yl)meth...)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248497(4-(2-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-indol-6-...)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248541((2-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-indol-6-yl...)
Affinity DataIC50:  12.7nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Howard University

Curated by ChEMBL
LigandPNGBDBM50021437(5-Ethyl-5-phenylbarbituric acid | 5-Phenyl-5-ethyl...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of [3H]BTX-B binding to neurotoxin site 2 of sodium channel of rat cerebral cortex synaptoneurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Howard University

Curated by ChEMBL
LigandPNGBDBM50101816(CHEBI:8107 | Dilabid | Dilantin | Dilantin-125 | D...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of [3H]BTX-B binding to neurotoxin site 2 of sodium channel of rat cerebral cortex synaptoneurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Howard University

Curated by ChEMBL
LigandPNGBDBM50031299(6-(2,3-Dichloro-phenyl)-[1,2,4]triazine-3,5-diamin...)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of [3H]BTX-B binding to neurotoxin site 2 of sodium channel of rat cerebral cortex synaptoneurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Howard University

Curated by ChEMBL
LigandPNGBDBM50003659(5H-dibenzo[b,f]azepine-5-carboxamide | CARBAMAZEPI...)
Affinity DataIC50:  1.31E+5nMAssay Description:Inhibition of [3H]BTX-B binding to neurotoxin site 2 of sodium channel of rat cerebral cortex synaptoneurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Howard University

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataIC50:  1.52E+5nMAssay Description:Inhibition of [3H]BTX-B binding to neurotoxin site 2 of sodium channel of rat cerebral cortex synaptoneurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Howard University

Curated by ChEMBL
LigandPNGBDBM50470610(CHEMBL340064)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of [3H]BTX-B binding to neurotoxin site 2 of sodium channel of rat cerebral cortex synaptoneurosomesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Howard University

Curated by ChEMBL
LigandPNGBDBM50470609(ADD-196022 | CHEMBL29740)
Affinity DataIC50:  4.89E+5nMAssay Description:Inhibition of [3H]BTX-B binding to neurotoxin site 2 of sodium channel of rat cerebral cortex synaptoneurosomesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed