Found 4 Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 1/2/3 subunit alpha' and Ligand = 'BDBM50031299'
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of [3H]saxitoxin binding to rat brain sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 1.14E+5nMAssay Description:Inhibition of [3H]BTX-B binding to neurotoxin site 2 of sodium channel of rat cerebral cortex synaptoneurosomesMore data for this Ligand-Target Pair
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour
Curated by ChEMBL
Institut Henri Beaufour
Curated by ChEMBL
Affinity DataIC50: 1.86E+5nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain sodium channelMore data for this Ligand-Target Pair