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Found 517 with Last Name = 'nai' and Initial = 'y'
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50083552(1,9-di{4-[5-amino(imino)methylbenzo[b]furan-2-ylca...)
Affinity DataKi:  0.0190nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50083561(1-{4-[5-amino(imino)methylbenzo[b]thiophen-2-ylcar...)
Affinity DataKi:  0.0280nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50083556(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  0.0290nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50083541(1-{4-[5-amino(imino)methyl-4,5,6,7-tetrahydrothien...)
Affinity DataKi:  0.0460nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50083548(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  0.0570nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50064089(4-hydroxymethyl-7,10-diisopropyl-8,10,13-trimethyl...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50217306(CHEMBL112049)
Affinity DataKi:  0.120nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375457(CHEMBL261476)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375451(CHEMBL408579)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262566((2S,3S)-3-[(1R)-6-Methoxy-1-methyl-1-trifluorometh...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]spiperone from NK1 receptor in human IM9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375452(CHEMBL262092)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375451(CHEMBL408579)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375457(CHEMBL261476)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM86441(CAS_3045225 | NSC_3045225 | YM348)
Affinity DataKi:  0.890nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50083549(1-{4-[5-amino(imino)methylbenzo[b]furan-2-ylcarbon...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of tryptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375458(CHEMBL406851)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50064089(4-hydroxymethyl-7,10-diisopropyl-8,10,13-trimethyl...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]- PDBu binding to peptide C, rat brain PKC gammaMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375900(CHEMBL259480)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85528(CAS_3045226 | NSC_3045226 | Ro 60-0175)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375454(CHEMBL261045)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM86441(CAS_3045225 | NSC_3045225 | YM348)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375447(CHEMBL403927)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280454((10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-3...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375459(CHEMBL264172)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375448(CHEMBL403926)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375899(CHEMBL406585)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375458(CHEMBL406851)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375460(CHEMBL256420)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375452(CHEMBL262092)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375903(CHEMBL262862)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375459(CHEMBL264172)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375900(CHEMBL259480)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375460(CHEMBL256420)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375454(CHEMBL261045)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375446(CHEMBL273163)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375455(CHEMBL404969)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM86441(CAS_3045225 | NSC_3045225 | YM348)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375905(CHEMBL405829)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50015677((S)-1-hydroxymethyl-2-octanoyloxy-ethyl ester | 1,...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50001915(1-(3-chlorophenyl)piperazine | CHEMBL478 | m-Chlor...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50180252((2S)-1-(6-methoxy-1H-indazol-1-yl)propan-2-amine |...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375455(CHEMBL404969)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM85528(CAS_3045226 | NSC_3045226 | Ro 60-0175)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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