Compile Data Set for Download or QSAR
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Found 96 with Last Name = 'nannei' and Initial = 'r'
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]AB-MECA from human recombinant A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]CCK-8 from human recombinant CCKA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  8nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323051(1-Biphenyl-3-yl-ethanone, O-(1-naphthylaminocarbon...)
Affinity DataIC50:  10nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323050(1-Biphenyl-3-yl-ethanone, O-(4-fluorophenylaminoca...)
Affinity DataIC50:  17nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323049(1-Biphenyl-3-yl-ethanone, O-(4-methoxyphenylaminoc...)
Affinity DataIC50:  28nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50212747((E)-1-(4-((5,6-dimethoxy-2-oxoindolin-3-ylidene)me...)
Affinity DataIC50:  50nMAssay Description:Inhibition of RET in mouse NIH3T3MEN2A cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323052(1-Biphenyl-3-yl-ethanone, O-(phenylaminocarbonyl)o...)
Affinity DataIC50:  69nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323042(1-(3'-Aminocarbonyl-biphenyl-3-yl)-ethanone, O-(ph...)
Affinity DataIC50:  84nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323047(1-Biphenyl-3-yl-ethanone, O-[(4-pentylphenyl)amino...)
Affinity DataIC50:  100nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  100nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323043(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(1-piperidi...)
Affinity DataIC50:  112nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323044(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(dodecylami...)
Affinity DataIC50:  116nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50212748(3-(4-hydroxybenzylidene)-5,6-dimethoxyindolin-2-on...)
Affinity DataIC50:  170nMAssay Description:Inhibition of RET in mouse NIH3T3MEN2A cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323057(1-(4-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50:  200nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50212745((E)-1-(4-((5,6-dimethoxy-2-oxoindolin-3-ylidene)me...)
Affinity DataIC50:  200nMAssay Description:Inhibition of RET in mouse NIH3T3MEN2A cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293352(CHEMBL551486 | N-Hydroxy-E-3-[4'-hydroxymethylbiph...)
Affinity DataIC50:  220nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323046(1-Biphenyl-3-yl-ethanone, O-(1-piperidinocarbonyl)...)
Affinity DataIC50:  220nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323048(1-Biphenyl-3-yl-ethanone, O-[(5-benzo[b]thiophenyl...)
Affinity DataIC50:  232nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293353(CHEMBL539156 | N-Hydroxy-E-3-[4-(4-hydroxyphenyl)-...)
Affinity DataIC50:  310nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293354(CHEMBL555906 | N-hydroxy-E-3-[4'-Hydroxybiphenyl-3...)
Affinity DataIC50:  320nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293355(CHEMBL538710 | N-Hydroxy-E-3-(4'-cyanobiphenyl-4-y...)
Affinity DataIC50:  330nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323058(1-Biphenyl-4-yl-ethanone, O-(1-naphthylaminocarbon...)
Affinity DataIC50:  401nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293356(CHEMBL561212 | N-Hydroxy-E-3-(4'-thiophen-2-yl-phe...)
Affinity DataIC50:  450nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293357(CHEMBL565140 | N-Hydroxy-E-3-[3'-chloro-4'-hydroxy...)
Affinity DataIC50:  460nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50212751((E)-1-(4-((5,6-dimethoxy-2-oxoindolin-3-ylidene)me...)
Affinity DataIC50:  580nMAssay Description:Inhibition of RET in mouse NIH3T3MEN2A cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293358(CHEMBL556332 | N-Hydroxy-E-3-(4'-hydroxybiphenyl-4...)
Affinity DataIC50:  590nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293359(5-(Biphenyl-4-yl)-pentanoic acid N-hydroxyamide | ...)
Affinity DataIC50:  720nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323059(1-Biphenyl-4-yl-ethanone, O-(phenylaminocarbonyl)o...)
Affinity DataIC50:  760nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293360(CHEMBL556532 | N-Hydroxy-E-3-(biphenyl-4-yl)-acryl...)
Affinity DataIC50:  820nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323056(1-[4-(cyclohexyl)-phenyl]-ethanone,O-(1-naphthylam...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323055(1-[4-(2,5-Dimethyl-pyrrol-1-yl)-phenyl]-ethanone,O...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Università

Curated by ChEMBL
LigandPNGBDBM50323054(1-[2,2']Bithiophenyl-5-yl-ethanone, O-(1-naphthyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse brain FAAH assessed as conversion of [3H-ethanolamine]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293361(CHEMBL561209 | N-Hydroxy-E-3-(4'-methoxybiphenyl-4...)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293363(CHEMBL552750 | E,E-5-(4'-Cyano-biphenyl-4-yl)-pent...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293362(CHEMBL538713 | N-Hydroxy-E-3-[4-(1H-indol-5-yl)-ph...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293364(CHEMBL551151 | N-Hydroxy-3-(4'-hydroxybiphenyl-4-y...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293365(CHEMBL557066 | N-Hydroxy-E-3-(4'-chlorobiphenyl-4-...)
Affinity DataIC50:  1.86E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50212752((E)-N-(4-((5,6-dimethoxy-2-oxoindolin-3-ylidene)me...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of RET in mouse NIH3T3MEN2A cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293366(CHEMBL554573 | N-Hydroxy-E-3-(4-pyridin-4-yl-pheny...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293367(CHEMBL538712 | N-Hydroxy-E-3-[4'-dimethylaminobiph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293368(CHEMBL538967 | E,E-5-Biphenyl-4-yl-penta-2,4-dieno...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50293369(CHEMBL538364 | E,E-5-(4'-Methoxybiphenyl-4-yl)-pen...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of HDAC2 in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H](-)CGP 12177 from human recombinant beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]BRL 43694 from human recombinant 5HT3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5HT2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]CYP from 5HT1B receptor expressed in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50323040(1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]SQ 29548 from human recombinant TXA2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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