Affinity DataKi: 0.600nMAssay Description:Binding affinity to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Affinity to human Alpha-1B adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Affinity to human Alpha-1B adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Affinity to human Alpha-2C adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 66nMAssay Description:Affinity to human Alpha-1B adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Affinity to human Alpha-1B adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Affinity to human Alpha-1B adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair