Affinity DataKi: 0.230nMAssay Description:In vitro binding affinity at rat liver Angiotensin II receptor, type 1 was determined based on displacement of [125I]-Ang IIMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity at rat liver Angiotensin II receptor, type 1 was determined based on displacement of [125I]-Ang IIMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity at rat liver Angiotensin II receptor, type 1 was determined based on displacement of [125I]-Ang IIMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against Mouse vas deferens smooth muscleMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Inhibitory activity against Mouse vas deferens smooth muscleMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.510nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Binding affinity against delta receptor with [3H]-[p-Cl-Phe4]-DPDPEMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 0.790nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.860nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataIC50: 0.870nMAssay Description:Binding affinity against delta receptor with [3H]-[p-Cl-Phe4]-DPDPEMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.890nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibitory activity against Guinea pig ileum smooth muscleMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Guinea pig ileum smooth muscleMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Binding affinity against Opioid receptor mu 1 with [3H]-CTOPMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 22.4nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 141nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 264nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 325nMAssay Description:Displacement of [125I]echistatin from human integrin alpha5beta3 expressed in human A549 cells by binding assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 557nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair