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Found 270 with Last Name = 'nyberg' and Initial = 'f'
TargetType-1 angiotensin II receptor B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370684(CHEMBL1791349)
Affinity DataKi:  0.160nMpH: 7.4Assay Description:Binding affinity for angiotensin II receptor, type 1 in rat liver membrane using [125I]-Ang II as radioligand, in pH 7.4 Tris-HCl buffer for 2 hr at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370684(CHEMBL1791349)
Affinity DataKi:  0.180nMpH: 7.4Assay Description:Binding affinity for angiotensin II receptor, type 2 in pig uterus myometrium using [125I]-Ang II as radioligand, in pH 7.4 Tris-HCl buffer for 1.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50472361(CHEMBL406349)
Affinity DataKi:  0.190nMAssay Description:In vitro binding affinity against Angiotensin II receptor, type 1 from rat liver membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50015662(3-Amino-N-{1-[5-[2-[2-(1-carboxy-2-phenyl-ethylcar...)
Affinity DataKi:  0.230nMAssay Description:In vitro binding affinity at rat liver Angiotensin II receptor, type 1 was determined based on displacement of [125I]-Ang IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370575(CHEMBL1791308)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-Ang II from angiotensin II receptor type 2 in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436546(CHEMBL2397481)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370575(CHEMBL1791308)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-Ang II from angiotensin II receptor type 2 in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436546(CHEMBL2397481)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to substance P receptor (1 to 7 amino acids) binding site in rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to AT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]angiotensin 2 from AT2 receptor in pig uterus membrane after 1.5 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156167(CHEMBL361927 | butyl (5-isobutylthien-2-yl)sulfony...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228195(Angiotensin Ii | CHEBI:2719)
Affinity DataKi:  0.530nMAssay Description:In vitro binding affinity against Angiotensin II receptor, type 1 from rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50139783(Angiotensin II analogue | CHEMBL404996)
Affinity DataKi:  0.620nMAssay Description:Binding affinity for Angiotensin II receptor type 2 using [125I]- Ang II in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370375(CHEMBL268815)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370686(CHEMBL1791350)
Affinity DataKi:  0.700nMpH: 7.4Assay Description:Binding affinity for angiotensin II receptor, type 2 in pig uterus myometrium using [125I]-Ang II as radioligand, in pH 7.4 Tris-HCl buffer for 1.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50141059(CHEMBL289614 | L-162782 | N-Butyloxycarbonyl-4'-(2...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50199326(CHEMBL217673 | N-butyloxycarbonyl-2-(4-imidazol-1-...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50168428((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S)-4-({[(2S)-...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]-Ang II from angiotensin II receptor type 2 in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50208102(CHEMBL424755 | [4-NH2-Phe6] Ang II)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus myometrial membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370375(CHEMBL268815)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]-Ang II from angiotensin II receptor type 2 in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156176((2S,5R,7aR)-6-[2-((S)-Acetylamino)-3-methyl-butyry...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-Ang II from pig uterus myometrium angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50251514(CHEMBL480906 | N-Butoxycarbonyl-3-[4-(N-benzylcarb...)
Affinity DataKi:  1nMAssay Description:Displacement of [125]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125]Ang2 from AT1 receptor in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370375(CHEMBL268815)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-Ang II from pig uterus myometrium angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50188489((S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-p...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50188489((S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-p...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50308381(CHEMBL589979 | H-Arg-Pro-Lys-Pro-Gln-Gln-Phe-OH)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50308381(CHEMBL589979 | H-Arg-Pro-Lys-Pro-Gln-Gln-Phe-OH)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50308381(CHEMBL589979 | H-Arg-Pro-Lys-Pro-Gln-Gln-Phe-OH)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to substance P receptor (1 to 7 amino acids) binding site in rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50112097(CHEMBL266450 | analog of Angiotensin II with trans...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity at rat liver Angiotensin II receptor, type 1 was determined based on displacement of [125I]-Ang IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50112098(CHEMBL412045 | analog of Angiotensin II with cis v...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity at rat liver Angiotensin II receptor, type 1 was determined based on displacement of [125I]-Ang IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50195697((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S)-2-[(2S)-bu...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50276158(CHEMBL4127872)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50175584((S)-3-Amino-N-((S)-1-{1-[(S)-3-[2-[2-((S)-(S)-1-ca...)
Affinity DataKi:  1.85nMpH: 7.4Assay Description:Binding affinity for angiotensin II receptor, type 2 in pig uterus myometrium using [125I]-Ang II as radioligand, in pH 7.4 Tris-HCl buffer for 1.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  2nMAssay Description:Displacement of [125]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156178(CHEMBL216331 | c[Hcy3,5]Ang II)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]-Ang II from pig uterus myometrium angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370375(CHEMBL268815)
Affinity DataKi:  2.10nMAssay Description:Binding affinity for Angiotensin II receptor type 2 using [125I]- Ang II in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50141059(CHEMBL289614 | L-162782 | N-Butyloxycarbonyl-4'-(2...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125]Ang2 from AT1 receptor in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436553(CHEMBL2396664)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436553(CHEMBL2396664)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]SP1-7 from substance P receptor (1 to 7 amino acids) binding site in Sprague-Dawley rat spinal cord membranes after 60 mins by li...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50321070(CHEMBL1164560 | N-Butyloxycarbonyl-3-(4-pyrazole-1...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]angiotensin 2 from AT2 receptor in pig uterus membrane after 1.5 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50031942((6aR,9R)-4,6a,7-Trimethyl-4,6,6a,7,8,9-hexahydro-i...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [N-methyl-3H]LSD from human 5HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370576(CHEMBL1791309)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]-Ang II from angiotensin II receptor type 2 in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50251489(CHEMBL481089 | butyl 5-isobutyl-3-(4-(isopropylcar...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50370576(CHEMBL1791309)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]-Ang II from angiotensin II receptor type 2 in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50168424((3S)-3-amino-3-{[(1S)-1-{[(2S)-4-({[(2S)-1-[(2S)-2...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]-Ang II from angiotensin II receptor type 2 in pig uterus myometriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity at Angiotensin II receptor, type 2 in pig uterus myometrial membranes by [125I]-Ang II displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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