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Found 240 with Last Name = 'padia' and Initial = 'jk'
LigandPNGBDBM50073729((R)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50:  0.150nMAssay Description:In vitro inhibition of [125I]- Bolton Hunter CCK-8 binding to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50062005((S)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50:  0.150nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50062000(2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50:  0.990nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063665(CHEMBL9203 | N-(3-nitrophenyl)-2-[3,4-dihydro-3-[3...)
Affinity DataIC50:  1nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063640(CHEMBL9405 | N-(3-cyanobenzene)-2-[3,4-dihydro-3-[...)
Affinity DataIC50:  1.20nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063630(CHEMBL9188 | N-(3-ethylesterbenzoicacid)-2-[3,4-di...)
Affinity DataIC50:  1.5nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataIC50:  1.70nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50449747(CHEMBL2304062)
Affinity DataIC50:  1.70nMAssay Description:In vitro inhibition of [125I]- Bolton Hunter CCK-8 binding to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50063616(CHEMBL8890 | N-(3-tert-butylbenzoicacid)-2-[3,4-di...)
Affinity DataIC50:  1.90nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50281284(CHEMBL433384 | [[(S)-2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50:  2.30nMAssay Description:In vitro inhibition of [125I]- Bolton Hunter CCK-8 binding to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50063666(CHEMBL266557 | N-(3-ethylesterbenzoicacid)-2-[3,4-...)
Affinity DataIC50:  2.40nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50062003(CHEMBL138233 | [(R)-2-(1H-Indol-3-yl)-1-((R)-2-met...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50061997(CHEMBL138084 | [(R)-1-((1R,2R)-2-Hydroxy-cyclohexy...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50061994(CHEMBL138112 | [(R)-1-(2-Cyano-cyclohexylcarbamoyl...)
Affinity DataIC50:  3.5nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50062006(CHEMBL344882 | [(R)-1-((1R,2R)-2-Hydroxy-cyclohept...)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063636(CHEMBL9406 | N-(3-ethylesterbenzoicacid)-2-[3,4-di...)
Affinity DataIC50:  5nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063661(CHEMBL9267 | N-(3-ethylesterbenzoicacid)-2-[3,4-di...)
Affinity DataIC50:  5nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063650(CHEMBL275307 | N-(3-benzonitrile)-2-[3,4-dihydro-3...)
Affinity DataIC50:  5.80nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063644(CHEMBL276627 | N-(3-chlorophenyl)-2-[3,4-dihydro-3...)
Affinity DataIC50:  5.90nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50062001(CHEMBL344380 | [(R)-1-(2-Hydroxy-cyclohexylcarbamo...)
Affinity DataIC50:  6.20nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50061988(CHEMBL138657 | [(R)-1-((S)-1-Hydroxymethyl-2-pheny...)
Affinity DataIC50:  6.30nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50061993(CHEMBL337529 | [(R)-1-(3-Aza-bicyclo[3.2.2]non-3-y...)
Affinity DataIC50:  6.5nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063662(CHEMBL9534 | N-(3-Methoxy-phenyl)-N-[(methyl-pheny...)
Affinity DataIC50:  8nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063629(3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-b...)
Affinity DataIC50:  8nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063614(CHEMBL8954 | N-(3-trifluoromethylphenyl)-2-[3,4-di...)
Affinity DataIC50:  8nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  8.5nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50281277((R)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50:  9.30nMAssay Description:In vitro inhibition of [125I]- Bolton Hunter CCK-8 binding to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50063641(2-[2-(6-Bromo-1H-indol-3-yl)-ethyl]-3-(3-isopropox...)
Affinity DataIC50:  9.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50061990((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50:  9.30nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50006842(2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-3-(3-isopropox...)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50063645(CHEMBL9319 | N-(2-methoxyphenyl)-2-[3,4-dihydro-3-...)
Affinity DataIC50:  10nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063667(CHEMBL266120 | N-(3-methylphenyl)-2-[3,4-dihydro-3...)
Affinity DataIC50:  11nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50062008(CHEMBL342932 | [(R)-1-(Azepan-1-ylcarbamoyl)-2-(1H...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50454908(CHEMBL2112795)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063639(CHEMBL9524 | N-(3-ethylesterbenzoicacid)-2-[3,4-di...)
Affinity DataIC50:  14nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063649(CHEMBL9083 | N-(3-benzonitrile)-2-[3,4-dihydro-3-[...)
Affinity DataIC50:  14nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063652(CHEMBL8997 | N-(4-chlorophenyl)-2-[3,4-dihydro-3-[...)
Affinity DataIC50:  14nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063632(CHEMBL9422 | N-(4-Bromophenyl)-2-[3,4-dihydro-3-[3...)
Affinity DataIC50:  14nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063613(CHEMBL9291 | N-phenyl-2-[3,4-dihydro-3-[3-(1-methy...)
Affinity DataIC50:  15nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063627(CHEMBL9354 | N-(3-ethylesterbenzoicacid)-2-[3,4-di...)
Affinity DataIC50:  15nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063626(2-[2-(6-Bromo-1H-indol-3-yl)-ethyl]-3-(3-dimethyla...)
Affinity DataIC50:  16nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50449746(CHEMBL2304063)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of [125I]- Bolton Hunter CCK-8 binding to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50062012(CHEMBL344211 | [(R)-2-(1H-Indol-3-yl)-1-methyl-1-(...)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50061999(CHEMBL138952 | [(R)-1-(1-Benzyl-2-phenyl-ethylcarb...)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063648(CHEMBL8922 | N-(3-methoxyphenyl)-2-[3,4-dihydro-3-...)
Affinity DataIC50:  22nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50063630(CHEMBL9188 | N-(3-ethylesterbenzoicacid)-2-[3,4-di...)
Affinity DataIC50:  22nMAssay Description:Compound was evaluated for functional activity on Cholecystokinin type B receptor (CCK-B) receptor carried out on guinea pig stomach cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063646(3-[3-({(3-Methoxy-phenyl)-[(methyl-phenyl-carbamoy...)
Affinity DataIC50:  23nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063642(CHEMBL9311 | N-(4-methoxyphenyl)-2-[3,4-dihydro-3-...)
Affinity DataIC50:  25nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]-Bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50062015(CHEMBL139601 | [(R)-1-((1S,2S)-2-Hydroxy-cyclohept...)
Affinity DataIC50:  26nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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