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Found 100 with Last Name = 'pagani' and Initial = 'ed'
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470256(CHEMBL86200)
Affinity DataIC50:  22nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230226(CHEMBL144015)
Affinity DataIC50:  40nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230281(CHEMBL144682)
Affinity DataIC50:  48nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470255(CHEMBL87298)
Affinity DataIC50:  62nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470254(CHEMBL313940)
Affinity DataIC50:  67nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470258(CHEMBL87448)
Affinity DataIC50:  83nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50289368(Butane-1-sulfonic acid [3-(2,3-dibromo-5-oxo-5,6-d...)
Affinity DataIC50:  85nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230235(CHEMBL144395)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230227(CHEMBL356549)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230228(CHEMBL144154)
Affinity DataIC50:  160nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230229(CHEMBL144190)
Affinity DataIC50:  170nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230225(CHEMBL144713)
Affinity DataIC50:  230nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470257(CHEMBL87191)
Affinity DataIC50:  240nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM14362(6-(4-imidazol-1-ylphenyl)-5-methyl-4,5-dihydro-2H-...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289368(Butane-1-sulfonic acid [3-(2,3-dibromo-5-oxo-5,6-d...)
Affinity DataIC50:  290nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230231(CHEMBL556516)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM14363(3-(2-propoxyphenyl)-2,4,7,8,9-pentazabicyclo[4.3.0...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibition of phosphodiesterase (PDE V).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470259(CHEMBL313681)
Affinity DataIC50:  330nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM15296(6-methyl-2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridin...)
Affinity DataIC50:  360nMAssay Description:Inhibition of cAMP Phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470253(CHEMBL83014)
Affinity DataIC50:  430nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50289353(2,3-Dibromo-8-(4-methoxy-phenyl)-6H-imidazo[1,2-d]...)
Affinity DataIC50:  450nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230222(Medorinone | WIN-49016)
Affinity DataIC50:  550nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230237(CHEMBL357234)
Affinity DataIC50:  570nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230238(CHEMBL356805)
Affinity DataIC50:  600nMAssay Description:Inhibition of cAMP Phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289357(1-Butyl-3-[3-(2,3-dibromo-5-oxo-5,6-dihydro-imidaz...)
Affinity DataIC50:  650nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289360(2,3-Dibromo-8-phenyl-6H-imidazo[1,2-d][1,2,4]triaz...)
Affinity DataIC50:  770nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289361(Butane-1-sulfonic acid [4-(2,3-dibromo-5-oxo-5,6-d...)
Affinity DataIC50:  840nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289367(8-(4-Amino-phenyl)-2,3-dibromo-6H-imidazo[1,2-d][1...)
Affinity DataIC50:  910nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230223(CHEMBL144453)
Affinity DataIC50:  940nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230279(CHEMBL144706)
Affinity DataIC50:  960nMAssay Description:Inhibition of cAMP Phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289350(1-Butyl-3-[2-(2,3-dibromo-5-oxo-5,6-dihydro-imidaz...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289355(8-(2-Amino-phenyl)-2,3-dibromo-6H-imidazo[1,2-d][1...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289361(Butane-1-sulfonic acid [4-(2,3-dibromo-5-oxo-5,6-d...)
Affinity DataIC50:  1.02E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289353(2,3-Dibromo-8-(4-methoxy-phenyl)-6H-imidazo[1,2-d]...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289358(8-(3-Amino-phenyl)-2,3-dibromo-6H-imidazo[1,2-d][1...)
Affinity DataIC50:  1.15E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289357(1-Butyl-3-[3-(2,3-dibromo-5-oxo-5,6-dihydro-imidaz...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289354(CHEMBL426946 | N-[3-(2,3-Dibromo-5-oxo-5,6-dihydro...)
Affinity DataIC50:  1.22E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230239(CHEMBL343895)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230232(CHEMBL145429)
Affinity DataIC50:  1.42E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289367(8-(4-Amino-phenyl)-2,3-dibromo-6H-imidazo[1,2-d][1...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289362(2,3-Dibromo-8-cyclohexyl-6H-imidazo[1,2-d][1,2,4]t...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289361(Butane-1-sulfonic acid [4-(2,3-dibromo-5-oxo-5,6-d...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE V).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289356(1-Butyl-3-[4-(2,3-dibromo-5-oxo-5,6-dihydro-imidaz...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289366(CHEMBL366491 | N-[4-(2,3-Dibromo-5-oxo-5,6-dihydro...)
Affinity DataIC50:  1.82E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289360(2,3-Dibromo-8-phenyl-6H-imidazo[1,2-d][1,2,4]triaz...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289364(2,3-Dimethyl-8-phenyl-6H-imidazo[1,2-d][1,2,4]tria...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230224(CHEMBL147736)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289366(CHEMBL366491 | N-[4-(2,3-Dibromo-5-oxo-5,6-dihydro...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289351(2,3-Dibromo-8-phenyl-6H-imidazo[1,2-d][1,2,4]triaz...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE I).More data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50289358(8-(3-Amino-phenyl)-2,3-dibromo-6H-imidazo[1,2-d][1...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibition of phosphodiesterase (PDE III).More data for this Ligand-Target Pair
In DepthDetails Article
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