Affinity DataKi: 94nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
Affinity DataKi: 170nM ΔG°: -38.2kJ/mole IC50: 390nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
Affinity DataKi: 400nM ΔG°: -36.2kJ/mole IC50: 500nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
Affinity DataKi: 740nM ΔG°: -34.6kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nM ΔG°: -33.5kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
Affinity DataKi: 1.85E+3nM ΔG°: -32.4kJ/mole IC50: 890nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nM ΔG°: -30.2kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 5.90E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 6.20E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 7.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 8.10E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 1.39E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair