Compile Data Set for Download or QSAR
maximum 50k data
Found 84 with Last Name = 'pagano' and Initial = 'm'
TargetCathepsin B(Homo sapiens (Human))
Queen'S University of Belfast

LigandPNGBDBM81670(Peptidyl ene diones, COOEt)
Affinity DataKi:  94nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Queen'S University of Belfast

LigandPNGBDBM81671(Peptidyl ene diones, COOMe)
Affinity DataKi:  125nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM11319((5-oxo-5,6-dihydroindolo[1,2-a]quinazolin-7-yl)ace...)
Affinity DataKi:  170nM ΔG°:  -38.2kJ/mole IC50:  390nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM11323(4,5,6,7-tetrabromo-1H-1,2,3-benzotriazole | 4,5,6,...)
Affinity DataKi:  400nM ΔG°:  -36.2kJ/mole IC50:  500nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataKi:  740nM ΔG°:  -34.6kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCathepsin B(Homo sapiens (Human))
Queen'S University of Belfast

LigandPNGBDBM81670(Peptidyl ene diones, COOEt)
Affinity DataKi:  850nMAssay Description:Inhibition assay using peptidyl ene diones to inactivate human cathepsins B and L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataKi:  1.18E+3nM ΔG°:  -33.5kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
Affinity DataKi:  1.85E+3nM ΔG°:  -32.4kJ/mole IC50:  890nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM11324((2R,3R,4S,5R)-2-(5,6-dichloro-1H-1,3-benzodiazol-1...)
Affinity DataKi:  4.50E+3nM ΔG°:  -30.2kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185622(Apam-YET | CHEMBL210325)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185622(Apam-YET | CHEMBL210325)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185630(CHEMBL210871 | Pam-YDL)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185650(CHEMBL209568 | Pam-YET)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185630(CHEMBL210871 | Pam-YDL)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185649((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185650(CHEMBL209568 | Pam-YET)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185626((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185641(CHEMBL209984 | Pam-YNT)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185625(CHEMBL380390 | pAM-FKF)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185621((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  3.40E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185642((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185637((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185648((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  4.30E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185640((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  4.30E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185638((S)-2-{(S)-4-Carboxy-2-[(S)-2-hexanoylamino-3-(4-h...)
Affinity DataKi:  5.90E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185628((S)-2-{(S)-4-carboxy-2-[(S)-2-dodecanoylamino-3-(4...)
Affinity DataKi:  6.20E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185644((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185619((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  7.20E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185632((S)-2-{(S)-4-carboxy-2-[(S)-2-decanoylamino-3-(4-h...)
Affinity DataKi:  7.20E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185624((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  7.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185648((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185630(CHEMBL210871 | Pam-YDL)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185625(CHEMBL380390 | pAM-FKF)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185644((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185645((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185633((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185627((S)-2-{(S)-4-Carboxy-2-[(S)-3-(4-hydroxy-phenyl)-2...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185647((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185646(CHEMBL207452 | Pam-YKF)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185651((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185628((S)-2-{(S)-4-carboxy-2-[(S)-2-dodecanoylamino-3-(4...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185638((S)-2-{(S)-4-Carboxy-2-[(S)-2-hexanoylamino-3-(4-h...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185646(CHEMBL207452 | Pam-YKF)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185620(CHEMBL378655 | TVTFKF)
Affinity DataKi:  1.39E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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