TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma Research
Curated by PDSP Ki Database
Novartis Pharma Research
Curated by PDSP Ki Database
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Antagonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 802nMAssay Description:Antagonist activity at human S1P3R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 978nMAssay Description:Antagonist activity at human S1P5R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human S1P4R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human S1P2R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.670nMAssay Description:Competitive binding affinity to human S1P1R receptor expressed in CHO cell membranes by Schild plot analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at human S1P4R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P5R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair