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Found 13 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 3' and Ligand = 'BDBM82470'
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  5.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  5.62nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  9.54nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  9.55nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  11.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  13.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  13.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  63nMAssay Description:Binding affinity towards human Somatostatin receptor type 3 (sst3) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  107nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(RAT)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  115nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed