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Found 45 with Last Name = 'pereira' and Initial = 'ar'
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50359305(CHEMBL1928588)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50359305(CHEMBL1928588)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit alpha type-2(Saccharomyces cerevisiae s288c (Yeast))
University of California San Diego

LigandPNGBDBM154579((2S)-2-[(2S)-2-hexanamido-3-methylbutanamido]-N,N-...)
Affinity DataIC50:  1.20nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit alpha type-2(Saccharomyces cerevisiae s288c (Yeast))
University of California San Diego

LigandPNGBDBM154578(Carmaphycin A (1))
Affinity DataIC50:  1.5nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataIC50:  2.80nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataIC50:  9.5nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM15234((1R,3R,5S,9R,18S)-18-(methoxymethyl)-1,5-dimethyl-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
TargetProteasome subunit alpha type-2(Saccharomyces cerevisiae s288c (Yeast))
University of California San Diego

LigandPNGBDBM154578(Carmaphycin A (1))
Affinity DataIC50:  46.2nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332741((4aS,11cS)-9,10-Dihydroxy-4,4,11c-trimethyl-1,2,3,...)
Affinity DataIC50:  66nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332731((4aS,7R,12cS)-10,11-Dihydroxy-4,4,7,12c-tetramethy...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit alpha type-2(Saccharomyces cerevisiae s288c (Yeast))
University of California San Diego

LigandPNGBDBM154579((2S)-2-[(2S)-2-hexanamido-3-methylbutanamido]-N,N-...)
Affinity DataIC50:  112nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit alpha type-2(Saccharomyces cerevisiae s288c (Yeast))
University of California San Diego

LigandPNGBDBM154579((2S)-2-[(2S)-2-hexanamido-3-methylbutanamido]-N,N-...)
Affinity DataIC50:  165nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM12915(2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one |...)
Affinity DataIC50:  550nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332733((4'S,6R)-6'-bromo-2,2,4',6-tetramethyl-3',4'-dihyd...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332743((4aS,11cS)-9,10-Dihydroxy-4,4,11c-trimethyl-1,2,3,...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332731((4aS,7R,12cS)-10,11-Dihydroxy-4,4,7,12c-tetramethy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332742((4aS,11cS)-9-Hydroxy-10-methoxy-4,4,11c-trimethyl-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332743((4aS,11cS)-9,10-Dihydroxy-4,4,11c-trimethyl-1,2,3,...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332739((4aS,11cS)-6a,10-Dihydroxy-4,4,11c-trimethyl-1,3,4...)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332741((4aS,11cS)-9,10-Dihydroxy-4,4,11c-trimethyl-1,2,3,...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332736((4aS,7R,12cS)-4,4,7,12c-Tetramethyl-2,3,4,4a,5,6,7...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332738((4aS,7S,12cS)-4,4,7,12c-Tetramethyl-2,3,4,4a,5,6,7...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332738((4aS,7S,12cS)-4,4,7,12c-Tetramethyl-2,3,4,4a,5,6,7...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50359303(CHEMBL1928586)
Affinity DataIC50:  2.30E+3nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50359303(CHEMBL1928586)
Affinity DataIC50:  2.30E+3nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332740((4aS,11cS)-9,10-Dimethoxy-4,4,11c-trimethyl-1,2,3,...)
Affinity DataIC50:  2.64E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332732((4aS,7R,12cS)-9-Bromo-7a,11-dihydroxy-4,4,7,12c-te...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332740((4aS,11cS)-9,10-Dimethoxy-4,4,11c-trimethyl-1,2,3,...)
Affinity DataIC50:  5.12E+3nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332742((4aS,11cS)-9-Hydroxy-10-methoxy-4,4,11c-trimethyl-...)
Affinity DataIC50:  5.15E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332733((4'S,6R)-6'-bromo-2,2,4',6-tetramethyl-3',4'-dihyd...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332735((4aS,7R,12cS)-9-Bromo-4,4,7,12c-tetramethyl-2,3,4,...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332736((4aS,7R,12cS)-4,4,7,12c-Tetramethyl-2,3,4,4a,5,6,7...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332739((4aS,11cS)-6a,10-Dihydroxy-4,4,11c-trimethyl-1,3,4...)
Affinity DataIC50:  9.57E+3nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332734((4aS,7R,12cS)-9-Bromo-10-methoxy-4,4,7,12c-tetrame...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50359303(CHEMBL1928586)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332737((4aS,7R,12cS)-4,4,7,12c-Tetramethyl-2,3,4,4a,5,6,7...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332734((4aS,7R,12cS)-9-Bromo-10-methoxy-4,4,7,12c-tetrame...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50359304(CHEMBL1928587)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332732((4aS,7R,12cS)-9-Bromo-7a,11-dihydroxy-4,4,7,12c-te...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50359304(CHEMBL1928587)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332737((4aS,7R,12cS)-4,4,7,12c-Tetramethyl-2,3,4,4a,5,6,7...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50332735((4aS,7R,12cS)-9-Bromo-4,4,7,12c-tetramethyl-2,3,4,...)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cells by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit alpha type-2(Saccharomyces cerevisiae s288c (Yeast))
University of California San Diego

LigandPNGBDBM154579((2S)-2-[(2S)-2-hexanamido-3-methylbutanamido]-N,N-...)
Affinity DataIC50: >5.00E+4nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed