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Found 27 with Last Name = 'phife' and Initial = 'dw'
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287720(6,7-Dibromo-3-[(2S,5R)-5-(6-bromo-1H-indol-3-yl)-4...)
Affinity DataKi:  78nMAssay Description:Binding affinity against human Alpha-1b adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287720(6,7-Dibromo-3-[(2S,5R)-5-(6-bromo-1H-indol-3-yl)-4...)
Affinity DataKi:  80nMAssay Description:Compound was tested for its binding affinity towards Rat-1 cells stably expressing hamster Alpha-1b adrenergic receptor by displacing [125I]-HEAT (2-...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287718(6-Bromo-3-[4-(1H-indol-3-yl)-1H-imidazol-2-yl]-1H-...)
Affinity DataKi:  130nMAssay Description:Compound was tested for its binding affinity towards Rat-1 cells stably expressing hamster Alpha-1b adrenergic receptor by displacing [125I]-HEAT (2-...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50287720(6,7-Dibromo-3-[(2S,5R)-5-(6-bromo-1H-indol-3-yl)-4...)
Affinity DataKi:  138nMAssay Description:Binding affinity was determined against Alpha-1a adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287720(6,7-Dibromo-3-[(2S,5R)-5-(6-bromo-1H-indol-3-yl)-4...)
Affinity DataKi:  140nMAssay Description:Compound was tested for its binding affinity towards CHO cells expressing human Alpha-1a adrenergic receptor by displacing [125I]-HEAT (2-beta-(4-hyd...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287719(6-Bromo-3-[2-(1H-indol-3-yl)-1H-imidazol-4-yl]-1H-...)
Affinity DataKi:  170nMAssay Description:Compound was tested for its binding affinity towards Rat-1 cells stably expressing hamster Alpha-1b adrenergic receptor by displacing [125I]-HEAT (2-...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287723(6-bromo-3-[4-(6-bromo-1H-3-indolyl)-1H-2-imidazoly...)
Affinity DataKi:  520nMAssay Description:Compound was tested for its binding affinity towards Rat-1 cells stably expressing hamster Alpha-1b adrenergic receptor by displacing [125I]-HEAT (2-...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287719(6-Bromo-3-[2-(1H-indol-3-yl)-1H-imidazol-4-yl]-1H-...)
Affinity DataKi:  550nMAssay Description:Compound was tested for its binding affinity towards CHO cells expressing human Alpha-1a adrenergic receptor by displacing [125I]-HEAT (2-beta-(4-hyd...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287722(CHEMBL436760 | [4-(6-Bromo-1H-indol-3-yl)-1H-imida...)
Affinity DataKi:  740nMAssay Description:Compound was tested for its binding affinity towards Rat-1 cells stably expressing hamster Alpha-1b adrenergic receptor by displacing [125I]-HEAT (2-...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287718(6-Bromo-3-[4-(1H-indol-3-yl)-1H-imidazol-2-yl]-1H-...)
Affinity DataKi:  770nMAssay Description:Compound was tested for its binding affinity towards CHO cells expressing human Alpha-1a adrenergic receptor by displacing [125I]-HEAT (2-beta-(4-hyd...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287721((6-Hydroxy-1H-indol-3-yl)-[5-(1H-indol-3-yl)-1H-im...)
Affinity DataKi:  1.15E+3nMAssay Description:Compound was tested for its binding affinity towards Rat-1 cells stably expressing hamster Alpha-1b adrenergic receptor by displacing [125I]-HEAT (2-...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287723(6-bromo-3-[4-(6-bromo-1H-3-indolyl)-1H-2-imidazoly...)
Affinity DataKi:  2.14E+3nMAssay Description:Compound was tested for its binding affinity towards CHO cells expressing human Alpha-1a adrenergic receptor by displacing [125I]-HEAT (2-beta-(4-hyd...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287721((6-Hydroxy-1H-indol-3-yl)-[5-(1H-indol-3-yl)-1H-im...)
Affinity DataKi:  4.74E+3nMAssay Description:Compound was tested for its binding affinity towards Rat-1 cells stably expressing hamster alpha1b adrenergic receptor by displacing [125I]-HEAT (2-b...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287722(CHEMBL436760 | [4-(6-Bromo-1H-indol-3-yl)-1H-imida...)
Affinity DataKi:  1.26E+4nMAssay Description:Compound was tested for its binding affinity towards CHO cells expressing human Alpha-1a adrenergic receptor by displacing [125I]-HEAT (2-beta-(4-hyd...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286606((4aS,12bR)-11-Chloro-10-hydroxy-4,4,4a,12b-tetrame...)
Affinity DataIC50:  300nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50276581((+/-)-wiedendiol B | CHEMBL456619)
Affinity DataIC50:  600nMAssay Description:Compound was tested for CETP inhibition by a precipitation method to separate lipoproteins after incubation of radiolabeled HDL with LDL and CETP.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285079(4-Methoxy-3-((S)-2,5,5,8a-tetramethyl-3,4,4a,5,6,7...)
Affinity DataIC50:  1.00E+3nMAssay Description:Compound was tested for CETP inhibition by a precipitation method to separate lipoproteins after incubation of radiolabeled HDL with LDL and CETP.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50276581((+/-)-wiedendiol B | CHEMBL456619)
Affinity DataIC50:  5.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285079(4-Methoxy-3-((S)-2,5,5,8a-tetramethyl-3,4,4a,5,6,7...)
Affinity DataIC50:  5.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240865((4aS,6aS,12aR,12bS)-10-Hydroxy-4,4,6a,12b-tetramet...)
Affinity DataIC50:  6.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286611(5,5,9,10-tetramethyl-18-oxatetracyclo[8.8.0.01,6.0...)
Affinity DataIC50:  2.20E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286609(1-((4aS,12bR)-9,10-Diacetyl-4,4,4a,12b-tetramethyl...)
Affinity DataIC50:  2.30E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50242257(2-((1R,2S,4aS)-1,2,4a,5-Tetramethyl-1,2,3,4,4a,7,8...)
Affinity DataIC50:  2.50E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286610(13-methoxy-5,5,9,10-tetramethyl-18-oxatetracyclo[8...)
Affinity DataIC50:  4.60E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240866((-)-ilimaquinone | 2-Hydroxy-5-methoxy-3-((1R,2S,4...)
Affinity DataIC50:  1.00E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286608(CHEMBL60072 | Sulfircin analogue | Sulfuric acid m...)
Affinity DataIC50: >1.90E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286607((3bR,5aR,6S,7S,9aR,9bR)-7-Hydroxy-6-hydroxymethyl-...)
Affinity DataIC50:  1.96E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article