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Found 229 with Last Name = 'pugliese' and Initial = 'am'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257025(4-(cyclohexylamino)-2-phenylpyrido[2,3-e][1,2,4]tr...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257026(4-(cyclopentylamino)-2-phenylpyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]DPCPX from adenosine A1 receptor in bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM86709(Rec 27/0074)
Affinity DataKi:  0.890nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM86709(Rec 27/0074)
Affinity DataKi:  1.02nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM86710(Rec 27/0224)
Affinity DataKi:  1.05nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50086159(CHEMBL16488 | N-(1-Oxo-2-phenyl-1,2-dihydro-[1,2,4...)
Affinity DataKi:  1.47nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50271450(CHEMBL482701 | N-(2-(4-methoxyphenyl)-1-oxo-1,2-di...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  3.09nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256972(4-amino-2-phenylpyrido[2,3-e][1,2,4]triazolo[4,3-a...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DPCPX from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [125I]DPCPX from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256925(2-(4-methoxyphenyl)pyrido[2,3-e][1,2,4]triazolo[4,...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218930(1-benzyl-3-(2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4...)
Affinity DataKi:  3.35nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218923(CHEMBL390407 | N-(2-(4-methoxyphenyl)-2H-pyrazolo[...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218912(2-phenyl-N-(2-m-tolyl-2H-pyrazolo[3,4-c]quinolin-4...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50271536(4-benzylureido-1,2-dihydro-2-phenyl-1,2,4-triazolo...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [125I]DPCPX from adenosine A1 receptor in bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM86709(Rec 27/0074)
Affinity DataKi:  4.17nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218919(CHEMBL242424 | N-(2-m-tolyl-2H-pyrazolo[3,4-c]quin...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218917(CHEMBL242632 | N-(2-p-tolyl-2H-pyrazolo[3,4-c]quin...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218918(CHEMBL390408 | N-(2-(4-methoxyphenyl)-2H-pyrazolo[...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257074(CHEMBL474016 | N-(2-(4-methoxyphenyl)-1-oxo-1,2-di...)
Affinity DataKi:  4.54nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  4.57nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50271538(4-benzylureido-1,2-dihydro-6-nitro-2-phenyl-1,2,4-...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [125I]DPCPX from adenosine A1 receptor in bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50149357(2-(4-Methoxy-phenyl)-6-nitro-2H,5H-[1,2,4]triazolo...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50149358(4-Amino-6-nitro-2-phenyl-2H-[1,2,4]triazolo[4,3-a]...)
Affinity DataKi:  4.75nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM86709(Rec 27/0074)
Affinity DataKi:  5.13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50271497(4-bismethanesulfonylamino-2-phenyl-1,2,4-triazolo[...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218925(2-phenyl-N-(2-p-tolyl-2H-pyrazolo[3,4-c]quinolin-4...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM85833(N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]- ethyl]-N...)
Affinity DataKi:  5.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50189820(4-acetamido-1,2-dihydro-6-nitro-2-phenyl-1,2,4-tri...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218927(CHEMBL389318 | N-benzoyl-N-(2-phenyl-2H-pyrazolo[3...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50272033(CHEMBL502005 | N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50271580(4-(benzyloxy)-2-(4-methoxyphenyl)-[1,2,4]triazolo[...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257072(CHEMBL473839 | N-(1-oxo-2-phenyl-1,2-dihydropyrido...)
Affinity DataKi:  7.15nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218910(2-(3-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4(5...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257113(CHEMBL475026 | N-benzoyl-N-(2-(4-methoxyphenyl)-1-...)
Affinity DataKi:  7.75nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit&Aagrove

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  8.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257026(4-(cyclopentylamino)-2-phenylpyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218905(2,2-diphenyl-N-(2-phenyl-2H-pyrazolo[3,4-c]quinoli...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218915(CHEMBL397033 | N-(2-(4-methoxyphenyl)-2H-pyrazolo[...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218921(2,2-diphenyl-N-(2-p-tolyl-2H-pyrazolo[3,4-c]quinol...)
Affinity DataKi:  11.5nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257072(CHEMBL473839 | N-(1-oxo-2-phenyl-1,2-dihydropyrido...)
Affinity DataKi:  11.7nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218914(2-m-Tolyl-2,5-dihydro-pyrazolo[3,4-c]quinolin-4-on...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50271536(4-benzylureido-1,2-dihydro-2-phenyl-1,2,4-triazolo...)
Affinity DataKi:  12.3nMAssay Description:Displacement of [125I]DPCPX from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218910(2-(3-methoxyphenyl)-2H-pyrazolo[3,4-c]quinolin-4(5...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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