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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50271497'
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50271497(4-bismethanesulfonylamino-2-phenyl-1,2,4-triazolo[...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50271497(4-bismethanesulfonylamino-2-phenyl-1,2,4-triazolo[...)
Affinity DataEC50:  1.20E+4nMAssay Description:Antagonist activity at human adenosine A3 cells expressed in CHO cells assessed as inhibition of NECA-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed