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Found 29 with Last Name = 'raaka' and Initial = 'bm'
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232256(CHEMBL255074 | N-(3-phenoxybenzyl)-4-nitrobenzamid...)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at FFAR1 expressed in HEK-EM293 cells assessed as inhibition calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232261(3-(4-nitrophenoxy)-N-phenylbenzamide | CHEMBL43816...)
Affinity DataIC50:  5.30E+3nMAssay Description:Antagonist activity at FFAR1 expressed in HEK-EM293 cells assessed as inhibition calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189773(CHEMBL211129 | N-tert-butyl-5-amino-4-(2-fluoro-3-...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189777(CHEMBL212815 | N-tert-butyl-5-amino-4-(3-fluorophe...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189774(CHEMBL378091 | N-tert-butyl-5-amino-4-(3-hydroxyph...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189778(CHEMBL211405 | N-tert-butyl-5-amino-4-(3-methoxyph...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189779(CHEMBL377399 | N-tert-butyl-5-amino-4-(3-methoxyph...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyrotropin receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189778(CHEMBL211405 | N-tert-butyl-5-amino-4-(3-methoxyph...)
Affinity DataEC50:  6.50E+3nMAssay Description:Agonist activity at TSHR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GPR40 H86F mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human GPR40 H137A mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at human GPR40 H86A mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  6.80E+3nMAssay Description:Agonist activity at human GPR40 H137F mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  1.78E+4nMAssay Description:Agonist activity at human GPR40 N244A mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232250(2-(5-(naphthalen-1-ylmethylthio)-1,3,4-thiadiazol-...)
Affinity DataEC50:  1.80E+3nMAssay Description:Activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232251(3-(3-(benzyloxy)benzylamino)benzoic acid | CHEMBL2...)
Affinity DataEC50:  8.20E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232252(6-(5-(naphthalen-1-ylmethylene)-4-oxo-2-thioxothia...)
Affinity DataEC50:  1.22E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232253(CHEMBL252526 | methyl 2-(5-(benzylthio)-1,3,4-thia...)
Affinity DataEC50:  1.67E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232254(3-(4-(allyloxy)benzylamino)benzoic acid | CHEMBL25...)
Affinity DataEC50:  1.45E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232255(4-(benzo[d][1,3]dioxol-5-ylmethylamino)benzoic aci...)
Affinity DataEC50:  2.46E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232250(2-(5-(naphthalen-1-ylmethylthio)-1,3,4-thiadiazol-...)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232258(4-(4-oxo-5-(thiophen-2-ylmethylene)-2-thioxothiazo...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232257(4-(5-(4-fluorobenzylidene)-4-oxo-2-thioxothiazolid...)
Affinity DataEC50:  2.26E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232259(4-(4-benzoylbenzamido)benzoic acid | CHEMBL404008)
Affinity DataEC50:  1.61E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232249(6-(4-oxo-5-(thiophen-2-ylmethylene)-2-thioxothiazo...)
Affinity DataEC50:  6.60E+3nMAssay Description:Activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232260(4-((5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-ylt...)
Affinity DataEC50:  1.51E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232262(4-(5-(furan-2-ylmethylene)-4-oxo-2-thioxothiazolid...)
Affinity DataEC50:  1.68E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50232249(6-(4-oxo-5-(thiophen-2-ylmethylene)-2-thioxothiazo...)
Affinity DataEC50:  7.60E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189775(CHEMBL377769 | N-tert-butyl-5-amino-4-(2,3-dimetho...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189776(CHEMBL211871 | tert-butyl 5-amino-4-(3-methoxyphen...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed