Affinity DataKi: 4.90nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 176nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 231nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:Displacement of [3H]-R-PIA from recombinant human adenosine A1 receptor expressed in CHO cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.76E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.17E+3nMAssay Description:Displacement of [3H]-R-PIA from recombinant human adenosine A1 receptor expressed in CHO cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.53E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.86E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.15E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.31E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Displacement of [3H]CGP54626 from GABA-B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.49E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 9.20E+4nMAssay Description:Displacement of [3H]CGP54626 from GABA-B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.77E+5nMAssay Description:Displacement of [3H]CGP54626 from GABA-B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 8.11nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 17.3nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Alexander Technological Education Institute Of Thessaloniki
Curated by ChEMBL
Alexander Technological Education Institute Of Thessaloniki
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of ovine COX1 assessed as PGF2alpha production by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 22.1nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 56.7nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 56.7nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Inhibition of human AChE by Ellmans testMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Alexander Technological Education Institute Of Thessaloniki
Curated by ChEMBL
Alexander Technological Education Institute Of Thessaloniki
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant COX-2 assessed as PGF2alpha production by enzyme immunoassayMore data for this Ligand-Target Pair