TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of Cyclin-dependent kinase 2 (CDK2/cyclin A)More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 730nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 790nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of recombinant human rhinovirus protease 3C using fluorogenic-Dabcyl-KTSAVLQSGFRKME-Edan as substrate after 5 mins by FRET assayMore data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 2 (CDK2/cyclin A)More data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of recombinant human rhinovirus protease 3C using fluorogenic-Dabcyl-KTSAVLQSGFRKME-Edan as substrate after 5 mins by FRET assayMore data for this Ligand-Target Pair
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of human coxsackievirus B3 protease 3C expressed in Escherichia coli (BL21) using fluorogenic-Dabcyl-KEALFQGPPQFE-Edans as substrate after...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.39E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibitory activity against topo II-mediated decatenation of DNAMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibitory activity against topo II-mediated decatenation of DNAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.05E+4nMAssay Description:Inhibitory activity against DNA topoisomerase IIMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical
Curated by ChEMBL
Ildong Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 2 (CDK2/cyclin A)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 2 (CDK2/cyclin A)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 2 (CDK2/cyclin A)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 4 (CDK4/cyclin Dl)More data for this Ligand-Target Pair