Compile Data Set for Download or QSAR
maximum 50k data
Found 309 with Last Name = 'saito' and Initial = 'n'
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26214((3S,6S,10aS)-6-[(2S)-2-aminopropanamido]-N-(diphen...)
Affinity DataKi:  14nM ΔG°:  -44.4kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26223((3S,6S,10aS)-6-[(2S)-2-(methylamino)propanamido]-5...)
Affinity DataKi:  14nM ΔG°:  -44.4kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26225((3S,6S,10aS)-N-[(1R)-2,3-dihydro-1H-inden-1-yl]-6-...)
Affinity DataKi:  15nM ΔG°:  -44.2kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13211((3S,6S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
Affinity DataKi:  25nM ΔG°:  -43.0kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26218((3S,6S,10aS)-N-(diphenylmethyl)-6-[(2S)-2-(methyla...)
Affinity DataKi:  26nM ΔG°:  -42.9kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26215((3S,6S,10aS)-6-[(2S)-2-aminobutanamido]-N-(dipheny...)
Affinity DataKi:  39nM ΔG°:  -41.9kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26217((3S,6S,10aS)-6-[(2S)-2-aminobutanamido]-N-[(S)-nap...)
Affinity DataKi:  47nM ΔG°:  -41.4kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26212((3S,6S,9aS)-6-[(2S)-2-aminopropanamido]-N-(dipheny...)
Affinity DataKi:  60nM ΔG°:  -40.8kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
Affinity DataKi:  61nM ΔG°:  -40.8kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26219((3S,6S,10aS)-N-(diphenylmethyl)-6-[(2S)-2-(methyla...)
Affinity DataKi:  67nM ΔG°:  -40.5kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26211((3S,6S,10aS)-6-[(2S)-2-aminopropanamido]-N-benzyl-...)
Affinity DataKi:  100nM ΔG°:  -39.6kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC eta-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26210((3S,6S,9aS)-6-[(2S)-2-aminopropanamido]-N-benzyl-5...)
Affinity DataKi:  150nM ΔG°:  -38.6kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  216nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC delta-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM26224((3S,6S,10aS)-6-[(2S)-2-(methylamino)propanamido]-5...)
Affinity DataKi:  274nM ΔG°:  -37.1kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13142((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  290nM ΔG°:  -36.9kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC theta-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13210((3S,6S,8aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
Affinity DataKi:  350nM ΔG°:  -36.5kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057513((2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,4,5...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229773(1-hexyl-indolactam-V10 | CHEMBL401369)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC epsilon-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13200((2S,3S)-2-{[(2S)-1-[(2S)-2-[(2S)-2-aminopropanamid...)
Affinity DataKi:  580nM ΔG°:  -35.2kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 309 total ) | Next | Last >>
Jump to: