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Found 69 with Last Name = 'sancelme' and Initial = 'm'
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  700nMAssay Description:Inhibition of CDK2/Cyclin A (unknown origin)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM2581(3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)
Affinity DataIC50:  2.45E+3nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054428(13-(3,4-dihydroxy-6-hydroxymethyl-5-methoxytetrahy...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266465((Z/E)-(2S)-2-amino-5-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of CDK2/Cyclin A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266463((Z/E)-(2S)-2-amino-6-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of KDR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266466((Z/E)-(2S)-2-amino-5-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266463((Z/E)-(2S)-2-amino-6-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of cMet (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266465((Z/E)-(2S)-2-amino-5-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of cMet (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266466((Z/E)-(2S)-2-amino-5-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of cMet (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266465((Z/E)-(2S)-2-amino-5-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266465((Z/E)-(2S)-2-amino-5-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Ret (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266466((Z/E)-(2S)-2-amino-5-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Ret (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266463((Z/E)-(2S)-2-amino-6-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266465((Z/E)-(2S)-2-amino-5-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266466((Z/E)-(2S)-2-amino-5-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266465((Z/E)-(2S)-2-amino-5-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of KDR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266466((Z/E)-(2S)-2-amino-5-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of KDR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266463((Z/E)-(2S)-2-amino-6-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266465((Z/E)-(2S)-2-amino-5-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266466((Z/E)-(2S)-2-amino-5-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266463((Z/E)-(2S)-2-amino-6-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Ret (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266463((Z/E)-(2S)-2-amino-6-([(5-bromo-2-oxo-indolin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266464((Z/E)-(2S)-2-amino-6-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of KDR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266464((Z/E)-(2S)-2-amino-6-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266464((Z/E)-(2S)-2-amino-6-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of cMet (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266464((Z/E)-(2S)-2-amino-6-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Ret (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266464((Z/E)-(2S)-2-amino-6-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50266464((Z/E)-(2S)-2-amino-6-([(2-oxo-indolin-3-ylidene)me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054426(7-hydroxy-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50:  2.21E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054423(1,11-dichloro-13-(3,4-dihydroxy-6-hydroxymethyl-5-...)
Affinity DataIC50:  2.88E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054429(6-Hydroxy-12-(4-O-methyl-beta-D-glucopyrannosyl) -...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054425(6-amino-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrro...)
Affinity DataIC50:  4.35E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM2672(3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)
Affinity DataIC50:  4.47E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50060400(6-methyl-12-(3,4,5-trihydroxy-6-hydroxymethyltetra...)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054432(1,11-Dichloro-6-hydroxy-12-(4-O-methyl-beta-D-gluc...)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054434(6-(4-Semicarbazido)-6,7,12,13-tetrahydro-5,7-dioxo...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054422(6-hydroxy-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50:  7.92E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50060402(3,5-di(methylcarbonyloxy)-2-methylcarbonyloxymethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50060403(1,11-dichloro-12-(3,4-dihydroxy-6-hydroxymethyl-5-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054420(12-(3,4-dihydroxy-6-hydroxymethyl-5-methoxytetrahy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50162287((Rebeccamycin)1,11-dichloro-12-(3,4-dihydroxy-6-hy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50060401(6-methyl-12-(3,4,5-trihydroxy-6-methyltetrahydro-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50060404(12-(3,4-dihydroxy-6-hydroxymethyl-5-methoxytetrahy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054420(12-(3,4-dihydroxy-6-hydroxymethyl-5-methoxytetrahy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054418(1,11-dichloro-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054438(6-Amino-12-(4-O-methyl-beta-D-glucopyrannosyl) -6,...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054431(6-Formamido-12-(4-O-methyl-beta-D-glucopyrannosyl)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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