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Found 344 with Last Name = 'sarma' and Initial = 'k'
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165019(4-(Diethylamino)-2-butynyl alpha-phenylcyclohexane...)
Affinity DataKi:  0.950nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  6nMAssay Description:Ki value for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  6nMAssay Description:Ki value for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165008((+)-(R)-2-(alpha-(2-(Diisopropylamino)ethyl)benzyl...)
Affinity DataKi:  6.91nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165019(4-(Diethylamino)-2-butynyl alpha-phenylcyclohexane...)
Affinity DataKi:  6.97nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165008((+)-(R)-2-(alpha-(2-(Diisopropylamino)ethyl)benzyl...)
Affinity DataKi:  7.07nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165012(CHEMBL192065 | Hydroxy-diphenyl-acetic acid 4-(3-a...)
Affinity DataKi:  14nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165012(CHEMBL192065 | Hydroxy-diphenyl-acetic acid 4-(3-a...)
Affinity DataKi:  31nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165016(4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  34nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165016(4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  34nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165010(CHEMBL192537 | Cyclohexyl-hydroxy-phenyl-acetic ac...)
Affinity DataKi:  35nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  37nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165020(Bis-(4-fluoro-phenyl)-hydroxy-acetic acid 4-(3-aza...)
Affinity DataKi:  39nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165020(Bis-(4-fluoro-phenyl)-hydroxy-acetic acid 4-(3-aza...)
Affinity DataKi:  40nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165018(2-((1R,5S)-3-3-Aza-bicyclo[3.1.0]hex-3-yl-1-phenyl...)
Affinity DataKi:  50nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165010(CHEMBL192537 | Cyclohexyl-hydroxy-phenyl-acetic ac...)
Affinity DataKi:  72nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165016(4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  79nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165016(4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  79nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402859(CHEMBL2205591)
Affinity DataKi:  81.5nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165018(2-((1R,5S)-3-3-Aza-bicyclo[3.1.0]hex-3-yl-1-phenyl...)
Affinity DataKi:  105nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165022(4-Methyl-2-[3-((1R,5S)-1-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  118nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165022(4-Methyl-2-[3-((1R,5S)-1-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  221nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402858(CHEMBL2205592)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402864(CHEMBL2205615)
Affinity DataKi:  241nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165024(CHEMBL195169 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  291nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50380754(CHEMBL2017853)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli using para-nitrophenyl phosphate as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402863(CHEMBL2205616)
Affinity DataKi:  347nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165013(CHEMBL194870 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  366nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50380753(CHEMBL2017852)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli using para-nitrophenyl phosphate as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402857(CHEMBL2205593)
Affinity DataKi:  444nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50380755(CHEMBL2017854)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli using para-nitrophenyl phosphate as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50380756(CHEMBL2017855)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli using para-nitrophenyl phosphate as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402859(CHEMBL2205591)
Affinity DataKi:  594nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50380751(CHEMBL2017850)
Affinity DataKi:  600nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli using para-nitrophenyl phosphate as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402857(CHEMBL2205593)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165024(CHEMBL195169 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  639nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165013(CHEMBL194870 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  736nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50380749(CHEMBL2017848)
Affinity DataKi:  800nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli using para-nitrophenyl phosphate as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402860(CHEMBL2205588)
Affinity DataKi:  899nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402861(CHEMBL2205584)
Affinity DataKi:  904nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165014(CHEMBL190459 | Cyclopentyl-hydroxy-(4-methoxy-phen...)
Affinity DataKi:  964nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma

Curated by ChEMBL
LigandPNGBDBM50402862(CHEMBL2205620)
Affinity DataKi:  999nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165011((1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-pheny...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165021(2-[3-((1R,5S)-1,5-Dimethyl-3-aza-bicyclo[3.1.0]hex...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165021(2-[3-((1R,5S)-1,5-Dimethyl-3-aza-bicyclo[3.1.0]hex...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165009((1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-pheny...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50380738(CHEMBL2017836)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human recombinant PTP1B expressed in Escherichia coli using para-nitrophenyl phosphate as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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