Affinity DataKi: 0.00400nMAssay Description:Binding affinity to angiotensin-converting enzyme (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.0100nMAssay Description:Binding affinity to human somatostatin receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Binding affinity to rat kidney neutral endopeptidaseMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.0800nMAssay Description:Binding affinity to rat kidney neutral endopeptidaseMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.110nMAssay Description:Binding affinity to angiotensin-converting enzyme in rabbit lung assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.180nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.380nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.380nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to neutral endopeptidase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.437nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.759nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 0.891nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 0.933nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 0.955nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 0.980nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity to insulin regulated aminopeptidase (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity to neutral endopeptidase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to angiotensin-converting enzyme (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.5nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to delta opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 4.5nMAssay Description:Binding affinity to angiotensin-converting enzyme in rabbit lung assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5nMAssay Description:Binding affinity to delta opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5nMAssay Description:Binding affinity to neutral endopeptidase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to angiotensin-converting enzyme (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >10nMAssay Description:Binding affinity to neutral endopeptidase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 12nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 15nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair