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Found 277 with Last Name = 'sejer pedersen' and Initial = 'd'
TargetAngiotensin-converting enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50614466(CHEMBL5272537)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to angiotensin-converting enzyme (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))TBA
LigandPNGBDBM50103430(6-Amino-2-(3-(1H-indol-3-yl)-2-{[4-(2-oxo-2,3-dihy...)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to human somatostatin receptor type 2More data for this Ligand-Target Pair
TargetNeprilysin(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50614463(CHEMBL5283332)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity to rat kidney neutral endopeptidaseMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetNeprilysin(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50614462(CHEMBL5277842)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to rat kidney neutral endopeptidaseMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)TBA
LigandPNGBDBM50614462(CHEMBL5277842)
Affinity DataKi:  0.110nMAssay Description:Binding affinity to angiotensin-converting enzyme in rabbit lung assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614474(CHEMBL5274928)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614476(CHEMBL5280457)
Affinity DataKi:  0.380nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518984(CHEMBL4564189)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))TBA
LigandPNGBDBM50614468(CHEMBL5272269)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to neutral endopeptidase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518969(CHEMBL4514723)
Affinity DataKi:  0.437nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614472(CHEMBL5284501)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518981(CHEMBL4594173)
Affinity DataKi:  0.759nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataKi:  0.790nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518993(CHEMBL4527821)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518982(CHEMBL4462252)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518977(CHEMBL1160734)
Affinity DataKi:  0.933nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518973(CHEMBL4473518)
Affinity DataKi:  0.955nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614491(CHEMBL5278521)
Affinity DataKi:  0.980nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518969(CHEMBL4514723)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518968(CHEMBL4441975)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518978(CHEMBL4446394)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518968(CHEMBL4441975)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518977(CHEMBL1160734)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518979(CHEMBL4434772)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))TBA
LigandPNGBDBM50614477(CHEMBL5267589)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to insulin regulated aminopeptidase (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518979(CHEMBL4434772)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))TBA
LigandPNGBDBM50024102(((S)-2-Mercaptomethyl-3-phenyl-propionylamino)-ace...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to neutral endopeptidase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50614464(CHEMBL5281720)
Affinity DataKi:  2nMAssay Description:Binding affinity to angiotensin-converting enzyme (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614471(CHEMBL5266765)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518982(CHEMBL4462252)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614491(CHEMBL5278521)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to delta opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518974(CHEMBL4574652)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518984(CHEMBL4564189)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518993(CHEMBL4527821)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614492(CHEMBL5282233)
Affinity DataKi:  4.20nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)TBA
LigandPNGBDBM50614463(CHEMBL5283332)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to angiotensin-converting enzyme in rabbit lung assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614493(CHEMBL5277977)
Affinity DataKi:  5nMAssay Description:Binding affinity to delta opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetNeprilysin(Homo sapiens (Human))TBA
LigandPNGBDBM50614464(CHEMBL5281720)
Affinity DataKi:  5nMAssay Description:Binding affinity to neutral endopeptidase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518973(CHEMBL4473518)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518981(CHEMBL4594173)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))TBA
LigandPNGBDBM50614467(CHEMBL5279614)
Affinity DataKi:  10nMAssay Description:Binding affinity to angiotensin-converting enzyme (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetNeprilysin(Homo sapiens (Human))TBA
LigandPNGBDBM50614466(CHEMBL5272537)
Affinity DataKi: >10nMAssay Description:Binding affinity to neutral endopeptidase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518975(CHEMBL4450606)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614470(CHEMBL5279008)
Affinity DataKi:  13nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518976(CHEMBL4442559)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518972(CHEMBL1395661)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518974(CHEMBL4574652)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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