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Found 771 with Last Name = 'shen' and Initial = 'g'
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186746((2S)-2-AMINO-4-[(2R,3R)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  370nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186746((2S)-2-AMINO-4-[(2R,3R)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  430nMAssay Description:Inhibition of ferrous substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186747((2S)-2-AMINO-4-[(2R,3S)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  720nMAssay Description:Inhibition of ferrous substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186747((2S)-2-AMINO-4-[(2R,3S)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  720nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
TargetS-ribosylhomocysteine lyase(Escherichia coli (strain K12))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186747((2S)-2-AMINO-4-[(2R,3S)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of cobalt substituted Escherichia coli LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Vibrio harveyi (strain ATCC BAA-1116 / BB120))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186747((2S)-2-AMINO-4-[(2R,3S)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  9.70E+3nMAssay Description:Inhibition of cobalt substituted Vibrio harveyi LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186746((2S)-2-AMINO-4-[(2R,3R)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  1.06E+4nMAssay Description:Inhibition of zinc substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
TargetS-ribosylhomocysteine lyase(Escherichia coli (strain K12))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186746((2S)-2-AMINO-4-[(2R,3R)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  1.27E+4nMAssay Description:Inhibition of cobalt substituted Escherichia coli LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Vibrio harveyi (strain ATCC BAA-1116 / BB120))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186746((2S)-2-AMINO-4-[(2R,3R)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  1.28E+4nMAssay Description:Inhibition of cobalt substituted Vibrio harveyi LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186747((2S)-2-AMINO-4-[(2R,3S)-2,3-DIHYDROXY-3-N-HYDROXYC...)
Affinity DataKi:  1.96E+4nMAssay Description:Inhibition of zinc substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50142500((2S)-2-amino-4-(methylsulfanyl)butanoic acid | (S)...)
Affinity DataKi:  6.10E+4nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186742((2S)-2-amino-6-(N-formyl-N-hydroxylamino)hexanoic ...)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186743(CHEMBL383729 | S-ribosylcysteine)
Affinity DataKi:  7.00E+4nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186748((S)-2-amino-6-(2-mercaptoacetamido)hexanoic acid |...)
Affinity DataKi:  1.32E+5nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50148771((2R,3R)-N,2,3,4-TETRAHYDROXYBUTANAMIDE | (2R,4R)-2...)
Affinity DataKi:  1.47E+5nMAssay Description:Inhibition of ferrous substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186744((S)-2-amino-6-(3-mercaptopropanamido)hexanoic acid...)
Affinity DataKi:  1.55E+5nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50148771((2R,3R)-N,2,3,4-TETRAHYDROXYBUTANAMIDE | (2R,4R)-2...)
Affinity DataKi:  1.56E+5nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50186745((S)-2-amino-6-(4-mercaptobutanamido)hexanoic acid ...)
Affinity DataKi:  4.73E+5nMAssay Description:Inhibition of cobalt substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Vibrio harveyi (strain ATCC BAA-1116 / BB120))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50148771((2R,3R)-N,2,3,4-TETRAHYDROXYBUTANAMIDE | (2R,4R)-2...)
Affinity DataKi:  5.50E+5nMAssay Description:Inhibition of cobalt substituted Vibrio harveyi LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Escherichia coli (strain K12))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50148771((2R,3R)-N,2,3,4-TETRAHYDROXYBUTANAMIDE | (2R,4R)-2...)
Affinity DataKi:  7.20E+5nMAssay Description:Inhibition of cobalt substituted Escherichia coli LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-ribosylhomocysteine lyase(Bacillus subtilis)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50148771((2R,3R)-N,2,3,4-TETRAHYDROXYBUTANAMIDE | (2R,4R)-2...)
Affinity DataKi:  2.40E+6nMAssay Description:Inhibition of zinc substituted Bacillus subtilis LuxSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM14774(3-(cyclopropylmethoxy)-N-(3,5-dichloropyridin-4-yl...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of PDE4D (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267826(CHEMBL4096145)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267827(CHEMBL4076794)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267796(CHEMBL4098840)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267804(CHEMBL4070136)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267806(CHEMBL4071255)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM141473(US8921368, 192)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267852(CHEMBL4073562)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267828(CHEMBL4078773)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267852(CHEMBL4073562)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM141473(US8921368, 192)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267807(CHEMBL4060536)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267810(CHEMBL4068856)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267807(CHEMBL4060536)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267836(CHEMBL4105015)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267840(CHEMBL4062062)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267837(CHEMBL4060444)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267797(CHEMBL4080797)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267808(CHEMBL4087655)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267840(CHEMBL4062062)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267808(CHEMBL4087655)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267848(CHEMBL4091582)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267826(CHEMBL4096145)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267827(CHEMBL4076794)
Affinity DataIC50:  1nMAssay Description:Inhibition of GST-tagged JAK1 (unknown origin) after 3 hrs by Caliper assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28028(2-aminopyridine analogue, 7 | N-{4-[(2-amino-3-eth...)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed using baculovirus expressed GST-Met, and poly(Glu/Tyr) as the substrate in the presence of test compound. Dose response c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28030(2-aminopyridine analogue, 9 | N-{4-[(2-amino-3-chl...)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed using baculovirus expressed GST-Met, and poly(Glu/Tyr) as the substrate in the presence of test compound. Dose response c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267839(CHEMBL4076823)
Affinity DataIC50:  1nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50267848(CHEMBL4091582)
Affinity DataIC50:  1nMAssay Description:Inhibition of JAK3 (unknown origin) using CSKtide as substrate after 30 mins in presence of [gamma33P]ATP by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shanghai Hengrui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50331029((R,Z)-2-(5-Fluoro-2-oxo-1,2-dihydro-indol-3-yliden...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human VEGFR2 after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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