BindingDB PrimarySearch_ki

Found 1466 with Last Name = 'singh' and Initial = 'g'

Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50493145(CHEMBL2419149)

Ki: 0.00420nMAssay Description:Binding affinity to human adenosine A2A receptor expressed in HEK293T cells measured by radioligand binding assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Adenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50594655(CHEMBL5177144)

Ki: 0.0510nMAssay Description:Binding affinity to human adenosine A1A receptor measured by radioligand-based affinity assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Adenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50594654(CHEMBL5171044)

Ki: 0.0760nMAssay Description:Binding affinity to human adenosine A1A receptor measured by radioligand-based affinity assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615748(CHEMBL5272772)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615749(CHEMBL5271570)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615750(CHEMBL5268306)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615751(CHEMBL5273835)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615752(CHEMBL5284012)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615753(CHEMBL5275680)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615754(CHEMBL5290358)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615755(CHEMBL5284128)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615756(CHEMBL5282135)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615757(CHEMBL5270226)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615742(CHEMBL5269241)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615743(CHEMBL5283319)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615744(CHEMBL5276967)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615747(CHEMBL5280524)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615745(CHEMBL5272518)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM50615746(CHEMBL5291452)

Ki: 0.100nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50235055(CHEMBL4095355)

Ki: 0.200nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in HEK293 cells measured by cAMP functional assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50235053(CHEMBL4064207)

Ki: 0.25nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in HEK293 cells measured by cAMP functional assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Adenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50231590(CHEMBL4063997)

Ki: 0.280nMAssay Description:Antagonist activity at human adenosine A1A receptorMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Carbonic anhydrase 2(Homo sapiens (Human))TBA

PNG

BDBM50515815(CHEMBL4559197)

Ki: 0.400nMAssay Description:Inhibition of human recombinant CA2More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))TBA

PNG

BDBM50515838(CHEMBL4459675)

Ki: 0.400nMAssay Description:Inhibition of human recombinant CA2More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))TBA

PNG

BDBM50515806(CHEMBL4533252)

Ki: 0.400nMAssay Description:Inhibition of human recombinant CA2More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))TBA

PNG

BDBM50515807(CHEMBL4561870)

Ki: 0.400nMAssay Description:Inhibition of human recombinant CA2More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))TBA

PNG

BDBM50515839(CHEMBL4590447)

Ki: 0.400nMAssay Description:Inhibition of human recombinant CA2More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))TBA

PNG

BDBM50515811(CHEMBL4580659)

Ki: 0.400nMAssay Description:Inhibition of human recombinant CA2More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))TBA

PNG

BDBM50515814(CHEMBL4540711)

Ki: 0.400nMAssay Description:Inhibition of human recombinant CA2More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50594659(CHEMBL5182249)

Ki: 0.400nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cells incubated for 60 mins and measured by by scintillation coun...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Adenosine receptor A3(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50348176(CHEMBL1562432)

Ki: 0.441nMAssay Description:Antagonist activity at adenosine A3 receptor (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Amine oxidase [flavin-containing] A(Homo sapiens (Human))TBA

PNG

BDBM15613(4-chloro-N-(2-morpholin-4-ylethyl)benzamide | 4-ch...)

Ki: 0.5nMAssay Description:Inhibition of human MAO-A by spectrofluorimetric analysisMore data for this Ligand-Target Pair

PDB Reactome pathway
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Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)

Ki: 0.5nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50268232(8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phen...)

Ki: 0.553nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50018688(CHEMBL3291301)

Ki: 0.560nMAssay Description:Binding affinity to human adenosine A2A receptor measured by radioligand-based affinity assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Adenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50550813(CHEMBL1316674)

Ki: 0.700nMAssay Description:Antagonist activity at adenosine A1 receptor (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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3D Structure (crystal)

Adenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50003019(8-(Hexahydro-2,5-methano-pentalen-3a-yl)-1,3-dipro...)

Ki: 0.700nMAssay Description:Antagonist activity at adenosine A1 receptor (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Adenosine receptor A2b(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50232044(CHEMBL4083317)

Ki: 0.900nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in HEK293 cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(Homo sapiens (Human))
New York University

Curated by ChEMBL

PNG

BDBM50007400(4-Phenyl-1-(4-phenyl-butyl)-piperidine | 4-Phenyl-...)

Ki: 1nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]-haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair

PDB Reactome pathway
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Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50235052(CHEMBL4099688)

Ki: 1.10nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in HEK293 cells measured by cAMP functional assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Adenosine receptor A3(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50470471(CHEMBL4294479)

Ki: 1.20nMAssay Description:Binding affinity to human adenosine A3A receptorMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50254013(3-(4-Amino-3-methylbenzyl)-7-(2-furyl)-3H-[1,2,3]t...)

Ki: 1.30nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50594625(AB-928 | AB928 | Ab-928 | Ab928 | ETRUMADENANT | E...)

Ki: 1.5nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50594660(CHEMBL5203657)

Ki: 1.5nMAssay Description:Binding affinity to human adenosine A2A receptor expressed in HEK293 cells measured by radioligand based assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)

Ki: 1.60nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM493757(US10988455, Example 1(xcv))

Ki: 1.70nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Histamine H3 receptor(Homo sapiens (Human))
University Of Botswana

Curated by ChEMBL

PNG

BDBM50127832(3-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)

Ki: 2nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Adenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50231596(CHEMBL4074150)

Ki: 2nMAssay Description:Antagonist activity at human adenosine A1A receptorMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Adenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50231597(CHEMBL4102409)

Ki: 2nMAssay Description:Antagonist activity at human adenosine A1A receptorMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Adenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL

PNG

BDBM50231588(CHEMBL4084453)

Ki: 2nMAssay Description:Antagonist activity at human adenosine A1A receptorMore data for this Ligand-Target Pair

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Displayed 1 to 50 (of 1466 total ) | Next | Last >>

Filter my 1466 hits

Targets 82▿
- UDP-N-acetylenolpyruvoylglucosamine reductase 136
- Acetylcholinesterase 102
- Adenosine receptor A2a 100
- Prostaglandin G/H synthase 2 98
- Carbonic anhydrase 1 86
- Cholinesterase 86
- Carbonic anhydrase 2 84
- Xanthine dehydrogenase/oxidase 66
- Prostaglandin G/H synthase 1 64
- UDP-N-acetylglucosamine 1-carboxyvinyltransferase 55
- UDP-N-acetylmuramate--L-alanine ligase 48
- UDP-N-acetylmuramoylalanine--D-glutamate ligase 47
- Adenosine receptor A1 46
- Virion infectivity factor 44
- Adenosine receptor A3 39
- Cyclin-A2/Cyclin-dependent kinase 2 30
- Cyclin-T1/Cyclin-dependent kinase 9 30
- Amine oxidase [flavin-containing] B 29
- Amine oxidase [flavin-containing] A 25
- Sigma non-opioid intracellular receptor 1 24
- Carbonic anhydrase 9 24
- D(2) dopamine receptor 23
- cGMP-specific 3',5'-cyclic phosphodiesterase 16
- Polyunsaturated fatty acid lipoxygenase ALOX15 16
- Histamine H3 receptor 16
- Carbonic anhydrase 12 13
- Adenosine receptor A2b 12
- Carbonic anhydrase 4 8
- Aurora kinase A 7
- Polyunsaturated fatty acid 5-lipoxygenase 6
- Substance-K receptor 4
- Beta-secretase 1 4
- Substance-P receptor 4
- Cannabinoid receptor 1 3
- Chitinase B 3
- Cannabinoid receptor 2 3
- Epidermal growth factor receptor 3
- Dual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A 2
- High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A 2
- cGMP-dependent 3',5'-cyclic phosphodiesterase 2
- Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A 2
- High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A 2
- cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A 2
- cAMP-specific 3',5'-cyclic phosphodiesterase 4A 2
- Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha' 2
- Aromatase 2
- Bifunctional epoxide hydrolase 2 2
- Glutamate receptor ionotropic, NMDA 1/2A 2
- G-protein coupled receptor 55 2
- Phospholipase A2, membrane associated 2
- Androgen receptor 2
- Aurora kinase B 2
- High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A 2
- cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A 2
- Chitotriosidase-1 1
- Estrogen receptor 1
- UDP-N-acetylglucosamine 1-carboxyvinyltransferase 1 1
- Cytochrome P450 2C11 1
- Sigma intracellular receptor 2 1
- Histone acetyltransferase p300 1
- Cytochrome P450 1A1 1
- Cytochrome P450 1A2 1
- Kappa-type opioid receptor 1
- Cytochrome P450 3A7 1
- Cytochrome P450 2C9 1
- 5-hydroxytryptamine receptor 1A 1
- Delta-type opioid receptor 1
- Cytochrome P450 2A6 1
- Cytochrome P450 3A5 1
- Mu-type opioid receptor 1
- Cytochrome P450 3A4 1
- Steroid 17-alpha-hydroxylase/17,20 lyase 1
- Alpha-2B adrenergic receptor 1
- Acidic mammalian chitinase 1
- Cytochrome P450 1B1 1
- Alpha-2C adrenergic receptor 1
- 5-hydroxytryptamine receptor 2C 1
- 5-hydroxytryptamine receptor 2A 1
- D(1A) dopamine receptor 1
- Cytochrome P450 2C19 1
- Cytochrome P450 2D6 1
- Cytochrome P450 2B6 1
- ...
Publications 20▿
- Eur J Med Chem 227: (2022) 199
- Bioorg Med Chem Lett 16: 176-80 (2006) 112
- Eur J Med Chem 215: (2021) 104
- Bioorg Med Chem Lett 15: 2527-31 (2005) 74
- Bioorg Med Chem 46: (2021) 74
- Bioorg Med Chem Lett 13: 2591-4 (2003) 63
- J Med Chem 60: 9470-9489 (2017) 60
- Bioorg Med Chem 19: 1950-8 (2011) 54
- J Med Chem 61: 7929-7941 (2018) 49
- J Med Chem 59: 3920-34 (2016) 48
- J Med Chem 36: 3923-8 (1994) 47
- J Med Chem 59: 7677-82 (2016) 44
- Eur J Med Chem 46: 5237-57 (2011) 40
- J Med Chem 49: 6027-36 (2006) 38
- Bioorg Med Chem 23: 2121-8 (2015) 36
- J Med Chem 63: 12137-12155 (2020) 32
- Bioorg Med Chem Lett 24: 495-500 (2014) 12
- Eur J Med Chem 221: (2021) 12
- Bioorg Med Chem 38: (2021) 9
- Bioorg Med Chem Lett 23: 1945-8 (2013) 2
Institutions 14▿
- Wyeth Research 249
- Isf College Of Pharmacy 220
- Indian Institute Of Technology (Banaras Hindu University) 178
- Csir-Indian Institute of Integrative Medicine 60
- Guru Nanak Dev University 60
- Indo-Soviet Friendship College Of Pharmacy 54
- TBA 49
- New York University 47
- Sanford Burnham Prebys Medical Discovery Institute 44
- University Of Botswana 40
- Wyeth 38
- Csir-Indian Institute Of Integrative Medicine 36
- University Of Minnesota 32
- Astrazeneca 2
Affinity: 0.0042 to 3.0E+6 nM▿
- Ki 479
- IC50 980
- Kd 3
- EC50 4
- Affinity ≤ nM
Xtal structures: 24
Docked structures: 6
Catalog Cmpds: 86