TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataKi: 0.840nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.77nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]8-OH-DPAT from rat 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.42nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.47nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataKi: 4.84nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]-YM09151-2 from human cloned dopamine D4 receptor expressed in insect Sf9 cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataKi: 14.2nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 15.4nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-YM09151-2 from human cloned dopamine D4 receptor expressed in insect Sf9 cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataKi: 18.9nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 21.5nMAssay Description:Displacement of [3H]8-OH-DPAT from rat 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 27.6nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28.5nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28.5nMAssay Description:Displacement of [3H]neomonapride from dopamine D2 receptor in rat corpus striatumMore data for this Ligand-Target Pair
Affinity DataKi: 28.5nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]-YM09151-2 from human cloned dopamine D4 receptor expressed in insect Sf9 cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataKi: 40.4nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-YM09151-2 from human cloned dopamine D4 receptor expressed in insect Sf9 cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataKi: 70.4nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 71.9nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 72.3nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 73.8nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 79.6nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 97nMAssay Description:Displacement of [3H]neomonapride from dopamine D2 receptor in rat corpus striatumMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Displacement of [3H]-YM09151-2 from human cloned dopamine D4 receptor expressed in insect Sf9 cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataKi: 131nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 131nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 137nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataKi: 141nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database