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Found 164 with Last Name = 'tautermann' and Initial = 'cs'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0100nMAssay Description:Antagonist activity at human M3 receptor expressed in CHO cells assessed as inhibition of carbachol-induced response after 30 mins by AP-1-driven luc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to human M3 K523A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to human M3 R133A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to human M3 K213A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to human M3 D518A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0158nMAssay Description:Binding affinity to human M3 F225A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0158nMAssay Description:Binding affinity to human M3 E220A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0158nMAssay Description:Binding affinity to human M3 F222A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0158nMAssay Description:Binding affinity to wild type human M3 receptor expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity to human M3 E228A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity to human M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066861(BA-679-BR | Spiriva | Tiotropium Bromide | Tiotrop...)
Affinity DataKi:  0.0251nMAssay Description:Binding affinity to human M3 Q224A mutant expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50494453(CHEMBL3091665)
Affinity DataKi:  0.0501nMAssay Description:Binding affinity to wild type human M3 receptor expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50494455(CHEMBL3091664)
Affinity DataKi:  0.0631nMAssay Description:Binding affinity to wild type human M3 receptor expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50494458(CHEMBL3091667)
Affinity DataKi:  0.158nMAssay Description:Binding affinity to wild type human M3 receptor expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50494459(CHEMBL3091670)
Affinity DataKi:  0.316nMAssay Description:Binding affinity to wild type human M3 receptor expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50494454(CHEMBL3091666)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to wild type human M3 receptor expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50494457(CHEMBL3091668)
Affinity DataKi:  2nMAssay Description:Binding affinity to wild type human M3 receptor expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041091(CHEMBL3355965)
Affinity DataKi:  4nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041182(CHEMBL3355940)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041193(CHEMBL3355954)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041185(CHEMBL3355944)
Affinity DataKi:  4.80nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041192(CHEMBL3355953)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041198(CHEMBL3355960)
Affinity DataKi:  5nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50494456(CHEMBL3091669)
Affinity DataKi:  5nMAssay Description:Binding affinity to wild type human M3 receptor expressed in HEK293T cells up to 24 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041088(CHEMBL3355962)
Affinity DataKi:  5nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041150(CHEMBL3355932)
Affinity DataKi:  5.70nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041150(CHEMBL3355932)
Affinity DataKi:  10nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041090(CHEMBL3355964)
Affinity DataKi:  11nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041195(CHEMBL3355956)
Affinity DataKi:  16nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041181(CHEMBL3355939)
Affinity DataKi:  18nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041185(CHEMBL3355944)
Affinity DataKi:  24nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041203(CHEMBL3355942)
Affinity DataKi:  31nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041158(CHEMBL3355934)
Affinity DataKi:  32nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041174(CHEMBL3355938)
Affinity DataKi:  33nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041092(CHEMBL3355966)
Affinity DataKi:  34nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041174(CHEMBL3355938)
Affinity DataKi:  37nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041201(CHEMBL3355950)
Affinity DataKi:  38nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041186(CHEMBL3355945)
Affinity DataKi:  46nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041186(CHEMBL3355945)
Affinity DataKi:  48nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041182(CHEMBL3355940)
Affinity DataKi:  52nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041197(CHEMBL3355959)
Affinity DataKi:  54nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041157(CHEMBL3355933)
Affinity DataKi:  60nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041199(CHEMBL3355961)
Affinity DataKi:  60nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041191(CHEMBL3355952)
Affinity DataKi:  61nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041158(CHEMBL3355934)
Affinity DataKi:  62nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041090(CHEMBL3355964)
Affinity DataKi:  64nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041157(CHEMBL3355933)
Affinity DataKi:  65nMAssay Description:Displacement of [125J]-eotaxin-1 from mouse CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041184(CHEMBL3355943)
Affinity DataKi:  66nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50041190(CHEMBL3355951)
Affinity DataKi:  67nMAssay Description:Displacement of [125J]-eotaxin-1 from human CCR3 transfected in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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