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Found 147 with Last Name = 'terracciano' and Initial = 's'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171884(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy...)
Affinity DataKi:  0.0210nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171886(4-{2-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  2.14nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171888(4-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propoxy}...)
Affinity DataKi:  3.36nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171887(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy...)
Affinity DataKi:  4.13nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171885(4-{3-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  5.13nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171890(4-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-...)
Affinity DataKi:  7.12nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171894(4-{2-[4-(3-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-...)
Affinity DataKi:  27.1nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171891(4-[3-(4-Pyridin-2-yl-piperazin-1-yl)-propoxy]-4-az...)
Affinity DataKi:  30.3nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171893(4-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethoxy}...)
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171883(4-[3-(4-Pyrimidin-2-yl-piperazin-1-yl)-propoxy]-4-...)
Affinity DataKi:  49.5nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171883(4-[3-(4-Pyrimidin-2-yl-piperazin-1-yl)-propoxy]-4-...)
Affinity DataKi:  118nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171892(4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethoxy]-4-aza...)
Affinity DataKi:  382nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171889(4-[2-(4-Pyrimidin-2-yl-piperazin-1-yl)-ethoxy]-4-a...)
Affinity DataKi:  384nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171887(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy...)
Affinity DataKi:  423nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171888(4-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propoxy}...)
Affinity DataKi:  547nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171885(4-{3-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  670nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine D2 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171888(4-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propoxy}...)
Affinity DataKi:  733nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171885(4-{3-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171894(4-{2-[4-(3-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171892(4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethoxy]-4-aza...)
Affinity DataKi:  3.51E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171887(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy...)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171886(4-{2-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  4.01E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Università

Curated by ChEMBL
LigandPNGBDBM50171885(4-{3-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  4.51E+3nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171886(4-{2-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine D2 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171883(4-[3-(4-Pyrimidin-2-yl-piperazin-1-yl)-propoxy]-4-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171891(4-[3-(4-Pyridin-2-yl-piperazin-1-yl)-propoxy]-4-az...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171884(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine D2 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171890(4-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine D2 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Università

Curated by ChEMBL
LigandPNGBDBM50171890(4-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Università

Curated by ChEMBL
LigandPNGBDBM50171886(4-{2-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171890(4-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171893(4-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethoxy}...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171891(4-[3-(4-Pyridin-2-yl-piperazin-1-yl)-propoxy]-4-az...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171894(4-{2-[4-(3-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171893(4-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethoxy}...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171892(4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethoxy]-4-aza...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171890(4-{2-[4-(2-Chloro-phenyl)-piperazin-1-yl]-ethoxy}-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171886(4-{2-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171889(4-[2-(4-Pyrimidin-2-yl-piperazin-1-yl)-ethoxy]-4-a...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Università

Curated by ChEMBL
LigandPNGBDBM50171884(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171884(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171885(4-{3-[4-(3-Trifluoromethyl-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Università

Curated by ChEMBL
LigandPNGBDBM50171888(4-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propoxy}...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50171884(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propoxy...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Mashhad University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using BML-KI104 Fluor de Lys as substrate by fluorescence-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50317647((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-benzyl...)
Affinity DataIC50:  25nMAssay Description:Inhibition of full length HDAC3 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50317647((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-benzyl...)
Affinity DataIC50:  68nMAssay Description:Inhibition of full length HDAC1 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50405790(CHEMBL5284121)
Affinity DataIC50:  150nMAssay Description:Antagonist potency against carbachol induced inhibition of electrically stimulated guinea pig atria Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50317647((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-benzyl...)
Affinity DataIC50:  179nMAssay Description:Inhibition of full length HDAC2 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50464480(CHEMBL4282628)
Affinity DataIC50:  180nMAssay Description:Inhibition of mPGES1 in IL-1beta-stimulated human A549 cell microsomes using PGH2 as substrate assessed as reduction in PGE2 production preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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