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Found 56 with Last Name = 'tizot' and Initial = 'a'
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053877(Allyl-(9-allyl-2-{4-[2,2-bis-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053873(Allyl-(9-allyl-2-{4-[(2-methoxy-10,11-dihydro-5H-d...)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053900(Allyl-(9-allyl-2-{4-[(10,11-dihydro-5H-dibenzo[a,d...)
Affinity DataKi:  46nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053872(Allyl-(2-{4-[(10,11-dihydro-5H-dibenzo[a,d]cyclohe...)
Affinity DataKi:  48nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataKi:  58nMAssay Description:Inhibition of [3H]D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053880(Allyl-(9-allyl-6-{4-[(10,11-dihydro-5H-dibenzo[a,d...)
Affinity DataKi:  62nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053892(Allyl-(9-allyl-2-{4-[(6,7,8,9-tetrahydro-5H-benzoc...)
Affinity DataKi:  62nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053891((9-Allyl-2-{4-[(10,11-dihydro-5H-dibenzo[a,d]cyclo...)
Affinity DataKi:  84nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053885(Allyl-(9-allyl-2-{4-[(8-chloro-11-methyl-10,10-dio...)
Affinity DataKi:  87nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053888(CHEMBL85156 | N,N'-Diallyl-6-{4-[2,2-bis-(4-fluoro...)
Affinity DataKi:  89nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053871(Allyl-(9-allyl-6-{4-[(5H-dibenzo[a,d]cyclohepten-5...)
Affinity DataKi:  90nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053896(Allyl-(9-allyl-6-{4-[(6,11-dihydro-dibenzo[b,e]oxe...)
Affinity DataKi:  93nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053895(Allyl-(9-allyl-2-{4-[(2,3,4-trimethoxy-10,11-dihyd...)
Affinity DataKi:  99nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053893(Allyl-(9-allyl-6-{4-[(2-methoxy-10,11-dihydro-5H-d...)
Affinity DataKi:  110nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053870(Allyl-(9-allyl-2-{4-[(6,11-dihydro-dibenzo[b,e]oxe...)
Affinity DataKi:  120nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053875(Allyl-(9-allyl-2-{4-[(5H-dibenzo[a,d]cyclohepten-5...)
Affinity DataKi:  170nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053898(Allyl-(9-allyl-6-{4-[(8-chloro-11-methyl-10,10-dio...)
Affinity DataKi:  170nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053883(Allyl-(7-allyl-2-{4-[(10,11-dihydro-5H-dibenzo[a,d...)
Affinity DataKi:  200nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053884(Allyl-(1-allyl-6-{4-[(10,11-dihydro-5H-dibenzo[a,d...)
Affinity DataKi:  270nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053881(Allyl-(1-allyl-6-{4-[(2-methoxy-10,11-dihydro-5H-d...)
Affinity DataKi:  400nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053874(Allyl-{9-allyl-2-[4-(2,2,2-triphenyl-ethylamino)-p...)
Affinity DataKi:  410nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053890((1-Allyl-6-{4-[(2-methoxy-10,11-dihydro-5H-dibenzo...)
Affinity DataKi:  420nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053901(Allyl-(9-allyl-2-{4-[(naphthalen-1-ylmethyl)-amino...)
Affinity DataKi:  440nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053899(Allyl-(9-allyl-2-{4-[(10,10-dioxo-11-propyl-10,11-...)
Affinity DataKi:  490nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053889(Allyl-{9-allyl-2-[4-(6,11-dihydro-dibenzo[b,e]oxep...)
Affinity DataKi:  550nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053886((2-{4-[(10,11-Dihydro-5H-dibenzo[a,d]cyclohepten-5...)
Affinity DataKi:  560nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053878(Allyl-{9-allyl-6-[4-(10,11-dihydro-5H-dibenzo[a,d]...)
Affinity DataKi:  620nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053897(Allyl-{9-allyl-2-[4-(2,2-diphenyl-ethylamino)-pipe...)
Affinity DataKi:  630nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053876(Allyl-{9-allyl-2-[4-(10,11-dihydro-5H-dibenzo[a,d]...)
Affinity DataKi:  770nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053887(Allyl-(3-allyl-5-{4-[(10,11-dihydro-5H-dibenzo[a,d...)
Affinity DataKi:  860nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053882(CHEMBL340348 | [1-(9-Allyl-6-allylamino-9H-purin-2...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053882(CHEMBL340348 | [1-(9-Allyl-6-allylamino-9H-purin-2...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053879(Allyl-(9-allyl-6-{4-[(naphthalen-1-ylmethyl)-amino...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50053894(11-{[1-(9-Allyl-6-allylamino-9H-purin-2-yl)-piperi...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of [3H]-D-888 binding to L-type [Ca2+] channel of membranes from rat skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM6471(4-Anilino-7,8-dialkoxybenzo[g]quinoline-3-carbonit...)
Affinity DataIC50:  0.460nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM8((1R)-cyclohexane-1,2-diol | cis-1,2-cyclohexanedio...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM12255(AZD0530 | CHEMBL217092 | Compound 33 | N-(5-chloro...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50303801(CHEMBL571546 | N-benzyl-2-(5-(4-(2-morpholinoethox...)
Affinity DataIC50:  20nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342390(3-Amino-6-(2-dimethylamino-ethylamino)-4-phenylthi...)
Affinity DataIC50:  32nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342392(3-Amino-4-benzyl-6-(2-dimethylamino-ethylamino)-th...)
Affinity DataIC50:  40nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342393(3-Amino-6-(2-dimethylamino-ethylamino)-4-propylthi...)
Affinity DataIC50:  63nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342391(3-Amino-6-(2-dimethylamino-ethylamino)-4-phenylthi...)
Affinity DataIC50:  68nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342389(3-Amino-6-(2-dimethylamino-ethylamino)-4-phenylthi...)
Affinity DataIC50:  107nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342387(3-Amino-6-(2-dimethylamino-ethylamino)-4-methylthi...)
Affinity DataIC50:  230nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342388(3-Amino-6-(2-dimethylamino-ethylamino)-4-methylthi...)
Affinity DataIC50:  246nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342379(3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carbo...)
Affinity DataIC50:  269nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342386(3-Amino-4-methyl-6-trifluoromethyl-thieno[2,3-b]py...)
Affinity DataIC50:  330nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342381(3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carbo...)
Affinity DataIC50:  769nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342384(3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carbo...)
Affinity DataIC50:  840nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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