Compile Data Set for Download or QSAR
maximum 50k data
Found 130 with Last Name = 'trippodo' and Initial = 'nc'
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403254(CHEMBL51389)
Affinity DataIC50:  0.600nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403250(CHEMBL51780)
Affinity DataIC50:  1nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403253(CHEMBL301751)
Affinity DataIC50:  1.20nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403257(CHEMBL51438)
Affinity DataIC50:  1.70nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403261(CHEMBL51498)
Affinity DataIC50:  2.10nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403251(CHEMBL299441)
Affinity DataIC50:  2.20nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403258(CHEMBL301364)
Affinity DataIC50:  2.40nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403280(CHEMBL65545)
Affinity DataIC50:  3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403252(CHEMBL54036)
Affinity DataIC50:  3.10nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282861((S)-1-[(S)-2-((S)-2-Mercaptomethyl-3-phenyl-propio...)
Affinity DataIC50:  4nMAssay Description:Tested in vitro for inhibition of Angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403254(CHEMBL51389)
Affinity DataIC50:  4.40nMAssay Description:Tested in vitro for inhibition of Angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403261(CHEMBL51498)
Affinity DataIC50:  4.80nMAssay Description:Tested in vitro for inhibition of Angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048509((3S,6S,9aS)-6-((S)-2-Mercapto-3-phenyl-propionylam...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048505((S)-2-[(3S,7S)-3-((S)-2-Mercapto-3-phenyl-propiony...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50073120((4S,6S,9aS)-6-((S)-2-Mercapto-3-phenyl-propionylam...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against Angiotensin I converting enzyme (ACE) isolated from rabbit lung extract using hippuryl-L-histidyl-L-leucine (HHL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403255(CHEMBL50559)
Affinity DataIC50:  5.20nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403268(CHEMBL299875)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048512(CHEMBL299639 | [(S)-3-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403277(CHEMBL61566)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against angiotensin converting enzyme (ACE) in rat was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048512(CHEMBL299639 | [(S)-3-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of purified rat kidney Neutral endopeptidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50073118(CHEMBL319237 | [(S)-8-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against Angiotensin I converting enzyme (ACE) isolated from rabbit lung extract using hippuryl-L-histidyl-L-leucine (HHL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048512(CHEMBL299639 | [(S)-3-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Neutral Endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048512(CHEMBL299639 | [(S)-3-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  6.10nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403266(CHEMBL415932)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282861((S)-1-[(S)-2-((S)-2-Mercaptomethyl-3-phenyl-propio...)
Affinity DataIC50:  6.60nMAssay Description:Tested in vitro for inhibition of neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403274(CHEMBL66481)
Affinity DataIC50:  7nMAssay Description:In vitro inhibitory activity against angiotensin converting enzyme (ACE) in rat was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403266(CHEMBL415932)
Affinity DataIC50:  7nMAssay Description:Inhibition of Neutral Endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048504(CHEMBL148155 | [(3S,7R)-7-Allyl-3-((S)-2-mercapto-...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403280(CHEMBL65545)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory activity against angiotensin converting enzyme (ACE) in rat was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50073120((4S,6S,9aS)-6-((S)-2-Mercapto-3-phenyl-propionylam...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory activity against purified rat kidney neutral endopeptidase (NEP) using a fluorometric assay with dansyl-Gly-Phe-Arg as the substr...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048506(CHEMBL104054 | [(3S,7S)-3-((S)-2-Mercapto-3-phenyl...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048506(CHEMBL104054 | [(3S,7S)-3-((S)-2-Mercapto-3-phenyl...)
Affinity DataIC50:  8.20nMAssay Description:In vitro inhibitory activity against Angiotensin I converting enzyme (ACE) isolated from rabbit lung extract using hippuryl-L-histidyl-L-leucine (HHL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50073121(CHEMBL430484 | [(S)-6-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  9.60nMAssay Description:In vitro inhibitory activity against Angiotensin I converting enzyme (ACE) isolated from rabbit lung extract using hippuryl-L-histidyl-L-leucine (HHL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048515(CHEMBL345021 | [(3S,7R)-7-Isobutyl-3-((S)-2-mercap...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403278(CHEMBL62417)
Affinity DataIC50:  10nMAssay Description:In vitro inhibitory activity against angiotensin converting enzyme (ACE) in rat was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048500((4S,7S,10aS)-7-((S)-2-Mercapto-3-phenyl-propionyla...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048513(CHEMBL147043 | [(3S,7S)-3-((S)-2-Mercapto-3-phenyl...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048512(CHEMBL299639 | [(S)-3-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory activity against angiotensin converting enzyme (ACE) in rat was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403279(CHEMBL66254)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory activity against angiotensin converting enzyme (ACE) in rat was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048512(CHEMBL299639 | [(S)-3-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50073119(CHEMBL107747 | Gemopatrilat | [(S)-6-((S)-2-Mercap...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory activity against Angiotensin I converting enzyme (ACE) isolated from rabbit lung extract using hippuryl-L-histidyl-L-leucine (HHL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048512(CHEMBL299639 | [(S)-3-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  12nMAssay Description:Tested in vitro for inhibition of Angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048512(CHEMBL299639 | [(S)-3-((S)-2-Mercapto-3-phenyl-pro...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403259(CHEMBL298388)
Affinity DataIC50:  13nMAssay Description:Tested in vitro for inhibition of Angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403260(CHEMBL53879)
Affinity DataIC50:  13nMAssay Description:Tested in vitro for inhibition of Angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048502(CHEMBL343191 | [(3S,7R)-3-((S)-2-Mercapto-3-phenyl...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme isolated from rabbit lung extract.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403267(CHEMBL422944)
Affinity DataIC50:  14nMAssay Description:Inhibition of Neutral Endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403262(CHEMBL300016)
Affinity DataIC50:  14nMAssay Description:Inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403251(CHEMBL299441)
Affinity DataIC50:  14nMAssay Description:Tested in vitro for inhibition of Angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403275(CHEMBL304881)
Affinity DataIC50:  16nMAssay Description:In vitro inhibitory activity against angiotensin converting enzyme (ACE) in rat was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
Displayed 1 to 50 (of 130 total ) | Next | Last >>
Jump to: