Affinity DataKi: 0.0372nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0398nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
Affinity DataKi: 0.0955nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of (-)-[3H]vesamicol from human VAChT expressed in rat PC12 A123.7 cells after 20 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of [125I]ABN from human D3 receptor transfected in HEK-293 cell membrane after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.182nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity against thymidylate synthase from L1210 mouse leukemia cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.209nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.209nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of (-)-[3H]vesamicol from human VAChT expressed in rat PC12 A123.7 cells after 20 hrsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
Affinity DataKi: 0.234nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.234nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity against thymidylate synthase from L1210 mouse leukemia cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.372nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.372nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Displacement of [125I]ABN from human D3 receptor transfected in HEK-293 cell membrane after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Binding affinity against thymidylate synthase from L1210 mouse leukemia cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [125I]ABN from human D3 receptor transfected in HEK-293 cell membrane after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.525nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.562nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of N-terminal His-6-tagged recombinant Aurora 1 (62 to 344) (unknown origin) expressed in baculovirus expression system by radiometric ass...More data for this Ligand-Target Pair
Affinity DataKi: 0.617nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.660nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.770nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Binding affinity against thymidylate synthase from L1210 mouse leukemia cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Binding affinity against thymidylate synthase from L1210 mouse leukemia cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.780nMAssay Description:Displacement of (-)-[3H]vesamicol from human VAChT expressed in rat PC12 cell membrane after 20 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.870nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]ABN from human D3 receptor transfected in HEK-293 cell membrane after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:In vitro binding affinity towards Nicotinic acetylcholine receptor alpha7 using [125I]-alpha-Bungarotoxin in rat brainMore data for this Ligand-Target Pair