Affinity DataIC50: 23nMAssay Description:SPA assays were run in displacement mode using 30 nM [3H]-GW3965. Ligands were tested in 12-point dose-response curves starting at 20 uM. IC50 values...More data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:SPA assays were run in displacement mode using 30 nM [3H]-GW3965. Ligands were tested in 12-point dose-response curves starting at 20 uM. IC50 values...More data for this Ligand-Target Pair
Affinity DataIC50: 121nMAssay Description:SPA assays were run in displacement mode using 30 nM [3H]-GW3965. Ligands were tested in 12-point dose-response curves starting at 20 uM. IC50 values...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:SPA assays were run in displacement mode using 30 nM [3H]-GW3965. Ligands were tested in 12-point dose-response curves starting at 20 uM. IC50 values...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:SPA assays were run in displacement mode using 30 nM [3H]-GW3965. Ligands were tested in 12-point dose-response curves starting at 20 uM. IC50 values...More data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+3nMAssay Description:SPA assays were run in displacement mode using 30 nM [3H]-GW3965. Ligands were tested in 12-point dose-response curves starting at 20 uM. IC50 values...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 6.14E+4nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 9.30E+4nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 2.75E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.21E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.40E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.50E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.58E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.63E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.79E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.81E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.89E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 3.94E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 4.06E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 4.09E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 4.48E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad Industrial De Santander
Curated by ChEMBL
Universidad Industrial De Santander
Curated by ChEMBL
Affinity DataIC50: 4.78E+5nMAssay Description:Inhibition of AChE (unknown origin) by Ellman colorimetric methodMore data for this Ligand-Target Pair
Affinity DataEC50: 97nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 180nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 70nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 3.90E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 400nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 6.70E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 900nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 900nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 700nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 27nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 300nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 67nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair
Affinity DataEC50: 76nMpH: 7.2 T: 2°CAssay Description:FRET-based co-activator recruitment assay measures agonist activities in a 384-well plate format. Reaction mixture containing His-tagged hLXR, biotin...More data for this Ligand-Target Pair