Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
Universita Degli Studi Di Milano
Universita Degli Studi Di Milano
Affinity DataKi: 25nM ΔG°: -43.1kJ/mole IC50: 460nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
Universita Degli Studi Di Milano
Universita Degli Studi Di Milano
Affinity DataKi: 61nM ΔG°: -40.9kJ/mole IC50: 530nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Agonist activity at human alpha2C adrenoceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor mic...More data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 178nMAssay Description:Agonist activity at human alpha2C adrenoceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor mic...More data for this Ligand-Target Pair
Affinity DataKi: 234nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Displacement of [3H]epibatidine from rat rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 339nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 339nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 562nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Binding affinity to 5HT4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of GST-tagged Tankyrases 2 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-tagged Tankyrases 1 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
Universita Degli Studi Di Milano
Universita Degli Studi Di Milano
Affinity DataIC50: 49nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair