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Found 42 with Last Name = 'waksman' and Initial = 'g'
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50105264(2-(2-Benzyl-3-hydroxycarbamoyl-propionylamino)-pro...)
Affinity DataKi:  1.70nMAssay Description:50% inhibitory activity against enkephalinase purified from rat kidney with [3H]D-Ala2-Leu-enkephalin (20 nM) as substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50405292(CHEMBL2079630)
Affinity DataKi:  1.80nMAssay Description:50% inhibitory activity against enkephalinase purified from rat kidney with [3H]D-Ala2-Leu-enkephalin (20 nM) as substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50405292(CHEMBL2079630)
Affinity DataKi:  2.90nMAssay Description:Inhibitory activity against aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50105264(2-(2-Benzyl-3-hydroxycarbamoyl-propionylamino)-pro...)
Affinity DataKi:  3.80nMAssay Description:Inhibitory activity against aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025920((2-Hydroxycarbamoyl-3-phenyl-propionylamino)-aceti...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025917((2-Hydroxyaminomethyl-3-phenyl-propionylamino)-ace...)
Affinity DataIC50: >1nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50002035((2-Hydroxycarbamoyl-3-phenyl-propionylamino)-aceti...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025914(2-Benzyl-N-(benzylcarbamoyl-methyl)-3-(formyl-hydr...)
Affinity DataIC50:  1.20nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50002022((2-Benzyl-3-hydroxycarbamoyl-propionylamino)-aceti...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025913(CHEMBL16457 | [2-(Formyl-hydroxy-amino)-3-phenyl-p...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50002022((2-Benzyl-3-hydroxycarbamoyl-propionylamino)-aceti...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50020158((R,S)2-(2-Benzyl-3-hydroxycarbamoyl-propionylamino...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50025913(CHEMBL16457 | [2-(Formyl-hydroxy-amino)-3-phenyl-p...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21641(2-(2-benzyl-3-sulfanylpropanamido)acetic acid | CH...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50020158((R,S)2-(2-Benzyl-3-hydroxycarbamoyl-propionylamino...)
Affinity DataIC50:  7.10nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50025915(CHEMBL16622 | [2-Benzyl-3-(formyl-hydroxy-amino)-p...)
Affinity DataIC50:  8.5nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025915(CHEMBL16622 | [2-Benzyl-3-(formyl-hydroxy-amino)-p...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50002035((2-Hydroxycarbamoyl-3-phenyl-propionylamino)-aceti...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025918(2-(Formyl-hydroxy-amino)-N-[(3-methyl-butylcarbamo...)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025921(CHEMBL17040 | [2-Benzyl-3-(formyl-hydroxy-amino)-p...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025922(2-Benzyl-N*4*-hydroxy-N*1*-[(3-methyl-butylcarbamo...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025911(2-Benzyl-N-carboxymethyl-malonamic acid | CHEMBL17...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025912(2-Benzyl-N-(benzylcarbamoyl-methyl)-N'-hydroxy-mal...)
Affinity DataIC50:  750nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025923(2-Benzyl-3-(formyl-hydroxy-amino)-N-[(3-methyl-but...)
Affinity DataIC50:  800nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025924(3-Benzyl-N-carboxymethyl-succinamic acid | CHEMBL1...)
Affinity DataIC50:  800nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025919(2-Benzyl-N-hydroxy-N'-[(3-methyl-butylcarbamoyl)-m...)
Affinity DataIC50:  850nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482437(CHEMBL1214127)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482440(CHEMBL1213950)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482436(CHEMBL1213997)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482432(CHEMBL1214051)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482441(CHEMBL1213947)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482433(CHEMBL1214054)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482428(CHEMBL1214128)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482438(CHEMBL1213882)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482427(CHEMBL1214126)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482434(CHEMBL1214125)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482430(CHEMBL1213948)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482439(CHEMBL1213996)
Affinity DataIC50:  1.59E+5nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482429(CHEMBL1213883)
Affinity DataIC50:  1.67E+5nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482431(CHEMBL1213949)
Affinity DataIC50:  3.04E+5nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChaperone protein PapD(Escherichia coli)
Ume£

Curated by ChEMBL
LigandPNGBDBM50482435(CHEMBL1213881)
Affinity DataIC50: >8.00E+5nMAssay Description:Inhibition of Escherichia coli UTI89 PapD chaperon assessed as inhibition of biofilm formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed