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Found 1628 with Last Name = 'waser' and Initial = 'b'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50413477(CHEMBL475226)
Affinity DataKi:  1nMAssay Description:Displacement of [125I](R)-1-(3-iodophenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1Hbenzo[e][1,4]diazepin-3-yl)urea from human CCK2 receptor expresse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50261388(H-c(Cys3-Phe6-Phe7-DTrp8-Lys9-Thr10-Phe11-Cys14)-O...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50413478(CHEMBL515288)
Affinity DataKi:  3.72nMAssay Description:Displacement of [125I](S)-1-(3-iodophenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)urea from human CCK1 receptor express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  3.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  3.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  3.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50243516((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-4-{[(1S)-1...)
Affinity DataKi:  5.51nMAssay Description:Binding affinity to human cloned sst2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85725(Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8...)
Affinity DataKi:  6.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi:  6.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  7.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50261388(H-c(Cys3-Phe6-Phe7-DTrp8-Lys9-Thr10-Phe11-Cys14)-O...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50243515((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-amin...)
Affinity DataKi:  26nMAssay Description:Binding affinity to human cloned sst2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50261388(H-c(Cys3-Phe6-Phe7-DTrp8-Lys9-Thr10-Phe11-Cys14)-O...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85723(des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naph...)
Affinity DataKi:  39nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50261388(H-c(Cys3-Phe6-Phe7-DTrp8-Lys9-Thr10-Phe11-Cys14)-O...)
Affinity DataKi:  44nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50261388(H-c(Cys3-Phe6-Phe7-DTrp8-Lys9-Thr10-Phe11-Cys14)-O...)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50243515((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-amin...)
Affinity DataKi:  48nMAssay Description:Binding affinity to human cloned sst5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50243516((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-4-{[(1S)-1...)
Affinity DataKi:  50nMAssay Description:Binding affinity to human cloned sst3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50243516((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-4-{[(1S)-1...)
Affinity DataKi:  50nMAssay Description:Binding affinity to human cloned sst5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi:  56nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85724(des-AA 1,2,4,5,12,13[DAgl8(Me,2-naphthoyl)]-SS)
Affinity DataKi:  70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85723(des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naph...)
Affinity DataKi:  70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM50243515((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-amin...)
Affinity DataKi:  93nMAssay Description:Binding affinity to human cloned sst3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85727(des-AA 1,2,4,5,12,13[D-Cys3, D-Agl8(Me,2-naphthoyl...)
Affinity DataKi:  115nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85520(CAS_5311373 | L-796,778 | NSC_5311373)
Affinity DataKi:  127nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi:  165nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi:  173nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50413477(CHEMBL475226)
Affinity DataKi:  174nMAssay Description:Displacement of [125I](S)-1-(3-iodophenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)urea from human CCK1 receptor express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50413478(CHEMBL515288)
Affinity DataKi:  537nMAssay Description:Displacement of [125I](R)-1-(3-iodophenyl)-3-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1Hbenzo[e][1,4]diazepin-3-yl)urea from human CCK2 receptor expresse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi:  607nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85727(des-AA 1,2,4,5,12,13[D-Cys3, D-Agl8(Me,2-naphthoyl...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85723(des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naph...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85520(CAS_5311373 | L-796,778 | NSC_5311373)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85725(Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85723(des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naph...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85724(des-AA 1,2,4,5,12,13[DAgl8(Me,2-naphthoyl)]-SS)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85723(des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naph...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85728(des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) | des-AA ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85724(des-AA 1,2,4,5,12,13[DAgl8(Me,2-naphthoyl)]-SS)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85723(des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naph...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne

Curated by PDSP Ki Database
LigandPNGBDBM85520(CAS_5311373 | L-796,778 | NSC_5311373)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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