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Found 395 with Last Name = 'welch' and Initial = 'wm'
TargetGlutamate receptor 3(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50096326(6-{(E)-2-[3-(2-Chloro-phenyl)-6-fluoro-4-oxo-3,4-d...)
In DepthDetails ArticlePubMed
LigandPNGBDBM50222081(CHEMBL327654)
Affinity DataKi:  5.10nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  5.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50222052(CHEMBL329548)
Affinity DataKi:  6.20nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50015720((hyoscine)3-Hydroxy-2-phenyl-propionic acid 9-meth...)
In DepthDetails PubMed
LigandPNGBDBM50222056(CHEMBL94017)
Affinity DataKi:  10nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82217(CHEMBL284994 | CP-52003 | SERTRALINE | [4-(3,4-Dic...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50222051(CHEMBL90118)
Affinity DataKi:  11nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50130287((4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-biphenyl-...)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222052(CHEMBL329548)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222053(CHEMBL90752)
Affinity DataKi:  18nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50130287((4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-biphenyl-...)
Affinity DataKi:  19nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222053(CHEMBL90752)
Affinity DataKi:  21nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50222082(CHEMBL544315)
Affinity DataKi:  22nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222055(CHEMBL327906)
Affinity DataKi:  24nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86698(BENZTROPINE | CAS_132-17-2 | CHEMBL116590 | NSC_23...)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM112777(NORTRIPTYLINE | US8629135, SW-02)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor 3(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50096327((R)-3-(2-Chloro-phenyl)-2-[(E)-2-(6-diethylaminome...)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222083(CHEMBL90538)
Affinity DataKi:  26nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222047(CHEMBL316283)
Affinity DataKi:  26nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222055(CHEMBL327906)
Affinity DataKi:  26nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222047(CHEMBL316283)
Affinity DataKi:  28nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222083(CHEMBL90538)
Affinity DataKi:  28nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222048(CHEMBL540821)
Affinity DataKi:  32nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222051(CHEMBL90118)
Affinity DataKi:  32nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82217(CHEMBL284994 | CP-52003 | SERTRALINE | [4-(3,4-Dic...)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82217(CHEMBL284994 | CP-52003 | SERTRALINE | [4-(3,4-Dic...)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222056(CHEMBL94017)
Affinity DataKi:  35nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222050(CHEMBL92856)
Affinity DataKi:  41nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222056(CHEMBL94017)
Affinity DataKi:  44nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222049(CHEMBL90150)
Affinity DataKi:  46nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82216(CP-52002)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor 3(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM85710(CP-471236)
Affinity DataKi:  57nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82217(CHEMBL284994 | CP-52003 | SERTRALINE | [4-(3,4-Dic...)
Affinity DataKi:  58nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82217(CHEMBL284994 | CP-52003 | SERTRALINE | [4-(3,4-Dic...)
Affinity DataKi:  58nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  66nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222051(CHEMBL90118)
Affinity DataKi:  69nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222050(CHEMBL92856)
Affinity DataKi:  74nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222049(CHEMBL90150)
Affinity DataKi:  79nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222048(CHEMBL540821)
Affinity DataKi:  89nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222082(CHEMBL544315)
Affinity DataKi:  91nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM77970(3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11...)
Affinity DataKi:  99nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222052(CHEMBL329548)
Affinity DataKi:  102nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222054(CHEMBL94056)
Affinity DataKi:  110nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM77970(3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11...)
Affinity DataKi:  110nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50020712(10,11-dihydro-5-(gamma-dimethylaminopropylidene)-5...)
Affinity DataKi:  130nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222055(CHEMBL327906)
Affinity DataKi:  132nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataKi:  150nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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