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Found 54 with Last Name = 'wilce' and Initial = 'mc'
TargetBifunctional ligase/repressor BirA(Escherichia coli)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataKi:  87nMAssay Description:Inhibition of Escherichia coli recombinant BPL using 3H-biotin as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Adelaide

LigandPNGBDBM92383(Biotin triazole, 14)
Affinity DataKi:  90nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388931(CHEMBL2063402)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataKi:  182nMAssay Description:Inhibition of human recombinant BPL using 3H-biotin as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388933(CHEMBL2063403)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Adelaide

LigandPNGBDBM92378(Biotin triazole, 5)
Affinity DataKi:  1.17E+3nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Adelaide

LigandPNGBDBM92382(Biotin triazole, 13)
Affinity DataKi:  1.17E+3nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388934(CHEMBL2063404)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388927(CHEMBL2063398)
Affinity DataKi:  3.85E+3nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388932(CHEMBL2062535)
Affinity DataKi:  6.43E+3nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Adelaide

LigandPNGBDBM92381(Biotin triazole, 12)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Adelaide

LigandPNGBDBM92380(Biotin triazole, 11)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Adelaide

LigandPNGBDBM92384(Biotin triazole, 15)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Adelaide

LigandPNGBDBM92385(Biotin triazole, 16)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
University of Adelaide

LigandPNGBDBM92379(Biotin triazole, 10)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388935(CHEMBL2063405)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388928(CHEMBL2063399)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388930(CHEMBL2063401)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388929(CHEMBL2063400)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50334297(CHEMBL1642690 | methyl 5-(2-ethyl-6-isopropylpheny...)
Affinity DataKd:  5.76E+3nMAssay Description:Binding affinity to human GRB7 expressed in Escherichia coli BL21 (DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50334298(CHEMBL1642691 | methyl 3-(6-benzoyl-3-hydroxyquino...)
Affinity DataKd:  3.06E+3nMAssay Description:Binding affinity to human GRB7 expressed in Escherichia coli BL21 (DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50334299(CHEMBL1642692 | methyl 3-(6-benzoyl-3-hydroxyquino...)
Affinity DataKd:  1.72E+4nMAssay Description:Binding affinity to human GRB7 expressed in Escherichia coli BL21 (DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250518(CHEMBL4093671)
Affinity DataKd:  220nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250520(CHEMBL4095044)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to GST-tagged GRB7-SH2 (415 to 532 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) in 50 mM sodium phosphate buff...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250517(CHEMBL4072970)
Affinity DataKd:  270nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250519(CHEMBL4069253)
Affinity DataKd:  830nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250522(CHEMBL4083407)
Affinity DataKd:  7.81E+3nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250524(CHEMBL4078046)
Affinity DataKd:  830nMAssay Description:Binding affinity to GST-tagged GRB7-SH2 (415 to 532 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) in 50 mM sodium phosphate buff...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250523(CHEMBL4101397)
Affinity DataKd:  1.57E+4nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250518(CHEMBL4093671)
Affinity DataKd:  2.94E+3nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250519(CHEMBL4069253)
Affinity DataKd:  130nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250517(CHEMBL4072970)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to GST-tagged GRB7-SH2 (415 to 532 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) in 1 mM sodium phosphate buffe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250520(CHEMBL4095044)
Affinity DataKd:  1.81E+4nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250522(CHEMBL4083407)
Affinity DataKd:  3.03E+3nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50334296(CHEMBL1642689 | methyl 5-(3-acetylphenylamino)-3-(...)
Affinity DataKd:  7.12E+3nMAssay Description:Binding affinity to human GRB7 expressed in Escherichia coli BL21 (DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50334295(CHEMBL1642688 | methyl 5-(2-cyano-4-nitrophenylami...)
Affinity DataKd:  6.57E+3nMAssay Description:Binding affinity to human GRB7 expressed in Escherichia coli BL21 (DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50250523(CHEMBL4101397)
Affinity DataKd:  2.56E+3nMAssay Description:Binding affinity to human GST-tagged GRB7-SH2 domain (415 to 594 residues) expressed in Escherichia coli BL21(DE3) pLys after 60 to 80 secs in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124407(CHEMBL3623448)
Affinity DataKd:  3.47E+5nMAssay Description:Binding affinity to Grb7-SH2 domain (unknown origin) without using phosphate buffer by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124407(CHEMBL3623448)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to Grb7-SH2 domain (unknown origin) using 100 mM phosphate buffer by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50124407(CHEMBL3623448)
Affinity DataKd:  2.00E+5nMAssay Description:Binding affinity to GST-tagged Grb2-SH2 domain (58 to 160 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124407(CHEMBL3623448)
Affinity DataKd:  1.81E+4nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124407(CHEMBL3623448)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 350 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124407(CHEMBL3623448)
Affinity DataKd:  2.90E+3nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 50 mM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124407(CHEMBL3623448)
Affinity DataKd:  3.47E+5nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 10(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50124406(CHEMBL3623450)
Affinity DataKd:  4.20E+5nMAssay Description:Binding affinity to GST-tagged Grb10-SH2 domain (471 to 594 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50124406(CHEMBL3623450)
Affinity DataKd:  5.60E+5nMAssay Description:Binding affinity to GST-tagged Grb2-SH2 domain (58 to 160 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124406(CHEMBL3623450)
Affinity DataKd:  2.10E+3nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124406(CHEMBL3623450)
Affinity DataKd:  6.57E+3nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 50 mM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50124405(CHEMBL3623449)
Affinity DataKd:  4.40E+5nMAssay Description:Binding affinity to GST-tagged Grb2-SH2 domain (58 to 160 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 7(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50124405(CHEMBL3623449)
Affinity DataKd:  5.70E+3nMAssay Description:Binding affinity to GST-tagged Grb7-SH2 domain (415 to 532 amino acid residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using 20 mM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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