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Found 351 with Last Name = 'wolak' and Initial = 'jp'
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26831(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  2nMpH: 7.0 T: 2°CAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26840(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  2nMpH: 7.0 T: 2°CAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26857(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  2nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26847(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  2nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26843(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  2nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50275692(CHEMBL528989 | N-(1-(3-methoxypropyl)-5-((phenylam...)
Affinity DataIC50:  3nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274339(CHEMBL485607 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  3nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196941(CHEMBL246365 | N2-(2-chlorobenzyl)-N4-((3-(aminome...)
Affinity DataIC50:  3nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26854(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  3nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274045(3-[2-[2-(4-Cyano-phenyl)-2-oxo-ethyl]-5-(2-cyclohe...)
Affinity DataIC50:  3nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274470(CHEMBL485555 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274340(CHEMBL483403 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274669(CHEMBL485031 | N-(1-(3-(1H-imidazol-1-yl)propyl)-5...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274471(CHEMBL485556 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196932(CHEMBL392642 | N2-(2-(methylthio)benzyl)-N4-((4-(a...)
Affinity DataIC50:  5nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274246(CHEMBL485232 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  5nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274671(4-cyano-N-(5-(N-methylcyclohexanecarboxamido)-1-(3...)
Affinity DataIC50:  5nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196957(CHEMBL246175 | N2-(2-bromobenzyl)-N4-((4-(aminomet...)
Affinity DataIC50:  5nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26839(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  5nMpH: 7.0 T: 2°CAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26856(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  5nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274705(4-cyano-N-(5-(N-methylcyclohexanecarboxamido)-1-(3...)
Affinity DataIC50:  5nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274558(4-cyano-N-(5-(N-methylcyclohexanecarboxamido)-1-ph...)
Affinity DataIC50:  6nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196961(CHEMBL246174 | N2-(2-(trifluoromethylthio)benzyl)-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26844(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  6nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50275651(CHEMBL487357 | N-(5-((cyclohexyl(methyl)amino)meth...)
Affinity DataIC50:  6nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196936(CHEMBL246386 | N2-(2,5-dichlorobenzyl)-N4-((4-(ami...)
Affinity DataIC50:  7nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274709(CHEMBL458787 | N-(1-(3-amino-3-oxopropyl)-5-(N-eth...)
Affinity DataIC50:  7nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274005(CHEMBL516958 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  8nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196978(CHEMBL246183 | N2-(2,3-dichlorobenzyl)-N4-((4-(ami...)
Affinity DataIC50:  8nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26853(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  8nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26841(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  8nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274631(4-cyano-N-(1-(3-(methylamino)-3-oxopropyl)-5-(N-me...)
Affinity DataIC50:  9nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274338(CHEMBL483397 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  9nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274206(CHEMBL485565 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  10nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274247(CHEMBL485233 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  10nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26855(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  10nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26846(5-(2-amino-1,3-thiazol-4-yl)-N-[(2E)-5-[benzene(me...)
Affinity DataIC50:  10nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274341(CHEMBL520312 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  10nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196959(CHEMBL396929 | N2-(2-nitrobenzyl)-N4-((4-(aminomet...)
Affinity DataIC50:  11nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26845(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  11nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26813(CHEMBL460824 | N-[(2E)-5-[benzene(methyl)amido]-1-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196951(CHEMBL247979 | N2-(2-(trifluoromethyl)benzyl)-N4-(...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274392(CHEMBL484940 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  12nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26848(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  13nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196987(CHEMBL245912 | N2-(2,3-dimethylbenzyl)-N4-((4-(ami...)
Affinity DataIC50:  13nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM50274632(4-cyano-N-(1-(3-(dimethylamino)-3-oxopropyl)-5-(N-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26842(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  14nMAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26832(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  14nMpH: 7.0 T: 2°CAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM26828(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50:  14nMpH: 7.0 T: 2°CAssay Description:Kinase is purified as a GST-fusion protein. The kinase activity is measured using DELFIA which utilizes europium chelate-labeled anti-phosphotyrosine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196991(CHEMBL245977 | N2-(2-(difluoromethyl)benzyl)-N4-((...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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