Affinity DataKi: 2.94E+3nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften
Curated by ChEMBL
Institut FüR Biowissenschaften
Curated by ChEMBL
Affinity DataKi: 9.40E+3nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften
Curated by ChEMBL
Institut FüR Biowissenschaften
Curated by ChEMBL
Affinity DataKi: 1.37E+4nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften
Curated by ChEMBL
Institut FüR Biowissenschaften
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant VEGF-R2 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of recombinant ALK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 975nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant ALK assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.87E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Heinrich-Heine-Universitat
Curated by ChEMBL
Heinrich-Heine-Universitat
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant CDK4/CycD1More data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of recombinant IGF1R (unknown origin) using Poly (Glu,Tyr) 4:1 as substrate assessed as incorporation of [gamma-33P]-ATP into substrate by...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of recombinant B-RAF-V600E mutantMore data for this Ligand-Target Pair
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of recombinant ALK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.28E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
Affinity DataIC50: 2.48E+3nMAssay Description:Inhibition of recombinant CDK2/CycAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich-Heine-Universitat
Curated by ChEMBL
Heinrich-Heine-Universitat
Curated by ChEMBL
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of recombinant SRCMore data for this Ligand-Target Pair
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
Affinity DataIC50: 2.82E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.99E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.03E+3nMAssay Description:Inhibition of recombinant FAK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of recombinant IGF1RMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of wild type MET (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.15E+3nMAssay Description:Inhibition of recombinant IGF1RMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of recombinant IGF1R (unknown origin) using Poly (Glu,Tyr) 4:1 as substrate assessed as incorporation of [gamma-33P]-ATP into substrate by...More data for this Ligand-Target Pair
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of recombinant ALK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.44E+3nMAssay Description:Inhibition of recombinant PDGFRbetaMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.52E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.67E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.67E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair