Compile Data Set for Download or QSAR
maximum 50k data
Found 432 with Last Name = 'wray' and Initial = 'v'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institut FüR Biowissenschaften

Curated by ChEMBL
LigandPNGBDBM50030271(CHEMBL127872 | N-[2-(8H-6-Thia-3,4,8-triaza-benzo[...)
Affinity DataKi:  2.94E+3nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften

Curated by ChEMBL
LigandPNGBDBM10849(1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-d...)
Affinity DataKi:  9.40E+3nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften

Curated by ChEMBL
LigandPNGBDBM50030271(CHEMBL127872 | N-[2-(8H-6-Thia-3,4,8-triaza-benzo[...)
Affinity DataKi:  1.37E+4nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institut FüR Biowissenschaften

Curated by ChEMBL
LigandPNGBDBM10849(1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-d...)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institut FüR Biowissenschaften

Curated by ChEMBL
LigandPNGBDBM10847(1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dion...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institut FüR Biowissenschaften

Curated by ChEMBL
LigandPNGBDBM10847(1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dion...)
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  650nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  800nMAssay Description:Inhibition of recombinant VEGF-R2 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446566(CHEMBL3109401)
Affinity DataIC50:  970nMAssay Description:Inhibition of recombinant ALK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  975nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of recombinant ALK assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  1.87E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Heinrich-Heine-Universitat

Curated by ChEMBL
LigandPNGBDBM50480485(Altersolanol A | CHEBI:2615)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of recombinant CDK4/CycD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446566(CHEMBL3109401)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibition of recombinant IGF1R (unknown origin) using Poly (Glu,Tyr) 4:1 as substrate assessed as incorporation of [gamma-33P]-ATP into substrate by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  2.18E+3nMAssay Description:Inhibition of recombinant B-RAF-V600E mutantMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446564(CHEMBL3109404)
Affinity DataIC50:  2.19E+3nMAssay Description:Inhibition of recombinant ALK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  2.21E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  2.22E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50480485(Altersolanol A | CHEBI:2615)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50480482(Alterporriol G/H | CHEBI:65389)
Affinity DataIC50:  2.26E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50480484(Macrosporin)
Affinity DataIC50:  2.28E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  2.48E+3nMAssay Description:Inhibition of recombinant CDK2/CycAMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich-Heine-Universitat

Curated by ChEMBL
LigandPNGBDBM50480482(Alterporriol G/H | CHEBI:65389)
Affinity DataIC50:  2.74E+3nMAssay Description:Inhibition of recombinant SRCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  2.82E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  2.87E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50480484(Macrosporin)
Affinity DataIC50:  2.99E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446566(CHEMBL3109401)
Affinity DataIC50:  3.03E+3nMAssay Description:Inhibition of recombinant FAK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50480482(Alterporriol G/H | CHEBI:65389)
Affinity DataIC50:  3.07E+3nMAssay Description:Inhibition of recombinant IGF1RMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446564(CHEMBL3109404)
Affinity DataIC50:  3.12E+3nMAssay Description:Inhibition of wild type MET (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of recombinant IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446565(CHEMBL3109402)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of recombinant IGF1R (unknown origin) using Poly (Glu,Tyr) 4:1 as substrate assessed as incorporation of [gamma-33P]-ATP into substrate by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446565(CHEMBL3109402)
Affinity DataIC50:  3.38E+3nMAssay Description:Inhibition of recombinant ALK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.44E+3nMAssay Description:Inhibition of recombinant PDGFRbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50276157(Alternariol 5-O-Methyl Ether | CHEMBL483526)
Affinity DataIC50:  3.52E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.56E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50276157(Alternariol 5-O-Methyl Ether | CHEMBL483526)
Affinity DataIC50:  3.67E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.67E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 432 total ) | Next | Last >>
Jump to: