Affinity DataKi: 68nMAssay Description:Binding affinity towards human leukocyte elastase at 10e-8 MMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity towards human leukocyte elastase at 10e-7 MMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding affinity towards human leukocyte elastase at 10e-8 MMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibitory activity against human leukocyte elastase at 10e-7 MMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.510nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Functional inhibition of ET-1 induced [Ca2+] increase in human Girardi heart (hGH) cells, which express Endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.810nMAssay Description:Inhibitory activity against 125 I-labeled ET-1 binding to Endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.810nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.920nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity towards endothelin A receptor in porcine aortic smooth muscle membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Binding affinity towards Endothelin B receptor in human girardi heart cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against 125 I-labeled ET-1 binding to Endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against 125 I-labeled ET-1 binding to Endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Binding affinity towards endothelin A receptor in porcine aortic smooth muscle membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Binding affinity towards endothelin A receptor in porcine aortic smooth muscle membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity towards endothelin A receptor in porcine aortic smooth muscle membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibitory activity against 125 I-labeled ET-1 binding to Endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity towards endothelin A receptor in porcine aortic smooth muscle membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibitory activity against 125 I-labeled ET-1 binding to Endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Binding affinity towards endothelin A receptor in porcine aortic smooth muscle membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Binding affinity towards endothelin A receptor in porcine aortic smooth muscle membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Binding affinity towards Endothelin A receptor in human neuroblastoma-derived cell line SK-N-MC membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Binding affinity towards endothelin B receptor in porcine cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity towards Endothelin A receptor in human neuroblastoma-derived cell line SK-N-MC membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibitory activity of the compound against I-labeled ET-1 binding to Endothelin A receptorMore data for this Ligand-Target Pair