TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibitory activity against HIV-1 Protease was determinedMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Imperial College
Curated by ChEMBL
Imperial College
Curated by ChEMBL
Affinity DataKi: 620nMAssay Description:Inhibition of recombinant human C-terminal His-tagged SIRT2 (50 to 389 end residues) expressed in Escherichia coli using tubulin-K40 peptide in prese...More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to recombinant human CNT1 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity to recombinant human CNT3 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 5 mins by sci...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Binding affinity was evaluated for competitive inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Binding affinity to recombinant human CNT3 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 5 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Binding affinity to recombinant human CNT1 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 5.30E+3nMAssay Description:Binding affinity to recombinant human CNT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity to recombinant human ENT1 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Binding affinity to recombinant human ENT1 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Competitive inhibition of mushroom tyrosinase after 30 mins by Lineweaver-Burk double reciprocal plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Binding affinity to recombinant human CNT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Competitive inhibition of mushroom tyrosinase after 30 mins by Lineweaver-Burk double reciprocal plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+4nMAssay Description:Binding affinity to recombinant human CNT1 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 3.80E+4nMAssay Description:Competitive inhibition of mushroom tyrosinase after 30 mins by Lineweaver-Burk double reciprocal plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+4nMAssay Description:Binding affinity to recombinant human ENT1 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+4nMAssay Description:Competitive inhibition of mushroom tyrosinase after 30 mins by Lineweaver-Burk double reciprocal plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.06E+5nMAssay Description:Binding affinity to recombinant human ENT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 1.26E+5nMAssay Description:Binding affinity to recombinant human CNT3 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 5 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 1.89E+5nMAssay Description:Binding affinity to recombinant human ENT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 2.31E+5nMAssay Description:Binding affinity to recombinant human CNT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
Affinity DataKi: 2.42E+5nMAssay Description:Binding affinity to recombinant human ENT2 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 15 mins by sc...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.240nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.420nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.430nMAssay Description:Inhibition of c-Met in human EBC-1 cells assessed as reduction in cell proliferation after 72 hrs by SRB or MTT assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.460nMAssay Description:Inhibition of c-Met in human MKN45 cells assessed as reduction in cell proliferation after 72 hrs by SRB or MTT assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.460nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.490nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.590nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition of c-Met in human EBC-1 cells assessed as reduction in cell proliferation after 72 hrs by SRB or MTT assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Inhibition of c-Met in human EBC-1 cells assessed as reduction in cell proliferation after 72 hrs by SRB or MTT assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of His-tagged FGFR3 V555M mutant (unknown origin) expressed in insect cells using poly Glu-Tyr preincubated for 1 hr followed by substrate...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of TPR-MET in mouse BAF3 cells assessed as reduction in cell proliferation after 72 hrs by SRB or MTT assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of c-Met in human EBC-1 cells assessed as reduction in cell proliferation after 72 hrs by SRB or MTT assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Chinese Academy Of Sciences (Cas)
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair