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Found 2 Enz. Inhib. hit(s) with Target = 'Solute carrier family 28 member 3' and Ligand = 'BDBM50138530'
TargetSolute carrier family 28 member 3(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50138530((2R,3R,5R)-2-Hydroxymethyl-5-{6-[(R)-(tetrahydro-f...)
Affinity DataKi:  1.26E+5nMAssay Description:Binding affinity to recombinant human CNT3 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 5 mins by sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 28 member 3(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50138530((2R,3R,5R)-2-Hydroxymethyl-5-{6-[(R)-(tetrahydro-f...)
Affinity DataIC50:  2.00E+5nMAssay Description:Binding affinity to recombinant human CNT3 expressed in Saccharomyces cerevisiae assessed as inhibition of [3H]-uridine transport after 5 mins by sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed