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Found 636 with Last Name = 'zhou' and Initial = 'hb'
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Wuhan University School Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)
Affinity DataKi: <1nMAssay Description:Inhibition of FAM-Bid binding to human BCL2 expressed in Escherichia coli BL21 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Wuhan University School Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50201732(CHEMBL3929718)
Affinity DataKi:  5nMAssay Description:Inhibition of FAM-Bid binding to human BCL2 expressed in Escherichia coli BL21 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19455(4-(3-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-5,7-bis(...)
Affinity DataKi:  7nM ΔG°:  -42.6kJ/mole EC50:  90nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458884(CHEMBL4206798)
Affinity DataKi:  11nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458882(CHEMBL4213948)
Affinity DataKi:  13nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50094707(CHEMBL3589346)
Affinity DataKi:  22nMAssay Description:Binding affinity to human ER-alpha ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458888(CHEMBL4205342)
Affinity DataKi:  24nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50571106(CHEMBL4853580)
Affinity DataKi:  24nMAssay Description:Binding affinity to human ERalpha LBD assessed as inhibition constant measured after 2 hrs by microplate readerMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50094709(CHEMBL3589349)
Affinity DataKi:  25nMAssay Description:Binding affinity to human ER-alpha ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19454(4-[2-(4-hydroxyphenyl)-5,7-bis(trifluoromethyl)pyr...)
Affinity DataKi:  26nM ΔG°:  -39.7kJ/mole EC50:  6.00E+3nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50571112(CHEMBL4855392)
Affinity DataKi:  27nMAssay Description:Binding affinity to human ERalpha LBD assessed as inhibition constant measured after 2 hrs by microplate readerMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458902(CHEMBL4214125)
Affinity DataKi:  30nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458897(CHEMBL4206281)
Affinity DataKi:  35nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094742(CHEMBL3589358)
Affinity DataKi:  39nMAssay Description:Binding affinity to human ER-beta ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458905(CHEMBL4208076)
Affinity DataKi:  40nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458904(CHEMBL4203290)
Affinity DataKi:  41nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458909(CHEMBL4207109)
Affinity DataKi:  43nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19456(4-(3-{4-[2-(dimethylamino)ethoxy]phenyl}-5,7-bis(t...)
Affinity DataKi:  47nM ΔG°:  -38.3kJ/mole EC50:  1.00E+3nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM19454(4-[2-(4-hydroxyphenyl)-5,7-bis(trifluoromethyl)pyr...)
Affinity DataKi:  48nM ΔG°:  -38.3kJ/mole EC50:  600nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094707(CHEMBL3589346)
Affinity DataKi:  49nMAssay Description:Binding affinity to human ER-beta ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458902(CHEMBL4214125)
Affinity DataKi:  50nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094744(CHEMBL3589360)
Affinity DataKi:  50nMAssay Description:Binding affinity to human ER-beta ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19453(4-[3-phenyl-5,7-bis(trifluoromethyl)pyrazolo[1,5-a...)
Affinity DataKi:  51nM ΔG°:  -38.1kJ/molepH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458882(CHEMBL4213948)
Affinity DataKi:  51nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458886(CHEMBL4217406)
Affinity DataKi:  52nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458905(CHEMBL4208076)
Affinity DataKi:  53nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50571109(CHEMBL4855191)
Affinity DataKi:  54nMAssay Description:Binding affinity to human ERalpha LBD assessed as inhibition constant measured after 2 hrs by microplate readerMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094739(CHEMBL3589368)
Affinity DataKi:  56nMAssay Description:Binding affinity to human ER-beta ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50094747(CHEMBL3589350)
Affinity DataKi:  57nMAssay Description:Binding affinity to human ER-alpha ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571106(CHEMBL4853580)
Affinity DataKi:  57nMAssay Description:Binding affinity to human ERbeta LBD assessed as inhibition constant measured after 2 hrs by microplate readerMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458903(CHEMBL4218543)
Affinity DataKi:  60nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50094708(CHEMBL3589347)
Affinity DataKi:  60nMAssay Description:Binding affinity to human ER-alpha ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094735(CHEMBL3589363)
Affinity DataKi:  61nMAssay Description:Binding affinity to human ER-beta ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458892(CHEMBL4208593)
Affinity DataKi:  62nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458887(CHEMBL4212982)
Affinity DataKi:  62nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094748(CHEMBL3589353)
Affinity DataKi:  68nMAssay Description:Binding affinity to human ER-beta ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM19455(4-(3-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-5,7-bis(...)
Affinity DataKi:  71nM ΔG°:  -37.4kJ/mole EC50:  40nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094748(CHEMBL3589353)
Affinity DataKi:  71nMAssay Description:Binding affinity to human ERbeta LBD assessed as inhibition constant measured after 2 hrs by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50094746(CHEMBL3589348)
Affinity DataKi:  71nMAssay Description:Binding affinity to human ER-alpha ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458900(CHEMBL4205171)
Affinity DataKi:  73nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458897(CHEMBL4206281)
Affinity DataKi:  73nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50094748(CHEMBL3589353)
Affinity DataKi:  79nMAssay Description:Binding affinity to human ERalpha LBD assessed as inhibition constant measured after 2 hrs by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50094750(CHEMBL3589357)
Affinity DataKi:  81nMAssay Description:Binding affinity to human ER-alpha ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50094748(CHEMBL3589353)
Affinity DataKi:  81nMAssay Description:Binding affinity to human ER-alpha ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094749(CHEMBL3589355)
Affinity DataKi:  82nMAssay Description:Binding affinity to human ER-beta ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50571108(CHEMBL4870760)
Affinity DataKi:  84nMAssay Description:Binding affinity to human ERalpha LBD assessed as inhibition constant measured after 2 hrs by microplate readerMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Wuhan University School Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50201737(CHEMBL1962393)
Affinity DataKi:  85nMAssay Description:Inhibition of FAM-Bid binding to human MCL1 expressed in Escherichia coli BL21 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50094711(CHEMBL3589352)
Affinity DataKi:  87nMAssay Description:Binding affinity to human ER-beta ligand binding domain after 2 hrs by competitive fluorometric binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM50458898(CHEMBL4210525)
Affinity DataKi:  88nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Wuhan University School Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50201738(CHEMBL3957283)
Affinity DataKi:  90nMAssay Description:Inhibition of FAM-Bid binding to human BCL2 expressed in Escherichia coli BL21 after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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