Affinity DataKi: 43nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 93nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair