Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 52313,93082,93084,93086,93089,52313,93082,93084,93086,93089   

TargetGlucose-1-phosphate thymidylyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of St. Andrews

LigandPNGBDBM93086(Analogue of 1a, 8b)
Affinity DataIC50: 102nMAssay Description:Inhibition assay using glucose-1-phosphate thymidylyltransferase (RmlA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2013
Entry Details Article
PubMed
TargetGlucose-1-phosphate thymidylyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of St. Andrews

LigandPNGBDBM93089(Analogue of 1a, 12b)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition assay using glucose-1-phosphate thymidylyltransferase (RmlA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlucose-1-phosphate thymidylyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of St. Andrews

LigandPNGBDBM93082(Analogue of 1a, 5)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition assay using glucose-1-phosphate thymidylyltransferase (RmlA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2013
Entry Details Article
PubMed
TargetGlucose-1-phosphate thymidylyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of St. Andrews

LigandPNGBDBM93084(Analogue of 1a, 8f)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition assay using glucose-1-phosphate thymidylyltransferase (RmlA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlucose-1-phosphate thymidylyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of St. Andrews

LigandPNGBDBM52313(6-azanyl-5-(methylamino)-1-(phenylmethyl)pyrimidin...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition assay using glucose-1-phosphate thymidylyltransferase (RmlA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2013
Entry Details Article
PubMed
TargetZinc finger protein mex-5(Caenorhabditis elegans)
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM52313(6-azanyl-5-(methylamino)-1-(phenylmethyl)pyrimidin...)
Affinity DataEC50:  9.21E+4nMAssay Description:Broad Institute: MLPCN maternal gene expression Project ID: 2024 Keywords: Zinc finger, C. elegans, maternal gene expression, RNA-protein interac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2011
Entry Details
PCBioAssay
TargetPOsterior Segregation(Caenorhabditis elegans)
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM52313(6-azanyl-5-(methylamino)-1-(phenylmethyl)pyrimidin...)
Affinity DataEC50:  3.00E+5nMAssay Description:Broad Institute: MLPCN maternal gene expression Project ID: 2024 Keywords: Zinc finger, C. elegans, maternal gene expression, RNA-protein interac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2011
Entry Details
PCBioAssay