Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
Ki: 300nMpH: 7.0Assay Description:Standard assay conditions for the determination of kinetic constants used a fluorogenic peptide substrate, typically H-D-Ala-Leu-Lys-AMC, and were de...More data for this Ligand-Target Pair
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
Ki: 1.45E+4nMAssay Description:The assay uses baculovirus-expressed human cathepsin S and the boc-Val-Leu-Lys-AMC fluorescent substrate available from Bachem in a 384 well plate fo...More data for this Ligand-Target Pair
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
BDBM123100(US10723709, Example 4 | US11312693, Example 4 | US...)
Ki: 1.45E+4nMpH: 7.0Assay Description:Standard assay conditions for the determination of kinetic constants used a fluorogenic peptide substrate, typically H-D-Ala-Leu-Lys-AMC, and were de...More data for this Ligand-Target Pair